SCHEMBL10153293

SCHEMBL10153293

COC(=O)C1C(=O)N(OCc2ccccc2)C(=O)c2cc(NC(=O)c3ccccc3)ccc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.45
RPS6KA2 Q15349 2/20 0.44
RAB9A P51151 4/20 0.42
NPC1 O15118 3/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
NR1H4 Q96RI1 2/20 0.42
ACE2 Q9BYF1 1/20 0.41
KMT2A Q03164 5/20 0.41
MEN1 O00255 3/20 0.41
NLRP3 Q96P20 1/20 0.41
MAPT P10636 2/20 0.40
USP2 O75604 1/20 0.40
MAPK1 P28482 1/20 0.40
ESR2 Q92731 1/20 0.40
TAAR1 Q96RJ0 1/20 0.40
POLB P06746 1/20 0.40
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
MCL1 Q07820 1/20 0.40
CTDSP1 Q9GZU7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10153594 0.90 ACHE (0.45) ACHERAB9ANPC1SMN1; SMN2KMT2A
SCHEMBL10153995 0.88 GRM4 (0.44) RAB9ANPC1SMN1; SMN2MAPTKCNK9
SCHEMBL9959325 0.87 APP (0.42) ACHEKMT2AMEN1MAPTMAPK1
SCHEMBL10153644 0.87 ALDH1A1 (0.42) ACHERPS6KA2RAB9ANPC1SMN1; SMN2
SCHEMBL10153305 0.85 MEN1 (0.46) RAB9ANPC1SMN1; SMN2KMT2AMEN1
SCHEMBL10153698 0.83 ALDH1A1 (0.39) KMT2AMEN1MAPTUSP2
SCHEMBL9959247 0.83 ALDH1A1 (0.42) ACHESMN1; SMN2KMT2AMEN1MAPT
SCHEMBL9960564 0.83 TRPA1 (0.38) KMT2AMEN1MAPT
SCHEMBL10153686 0.82 MEN1 (0.46) RAB9ANPC1SMN1; SMN2KMT2AMEN1
SCHEMBL9958850 0.82 MEN1 (0.43) KMT2AMEN1MAPTMAPK1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085003-A1 2-HYDROXYISOQUINOLINE-1,3(2H,4H)-DIONES AND RELATED COMPOUNDS USEFUL AS HIV REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2012-06-28 WO disclosed