SCHEMBL10158064

SCHEMBL10158064

CCCOc1ccc(CC)c(Cl)c1N

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK2A1 P68400 2/20 0.45
MAPT P10636 6/20 0.45
ALDH1A1 P00352 3/20 0.45
KDM4E B2RXH2 3/20 0.45
POLB P06746 2/20 0.45
MEN1 O00255 1/20 0.45
USP2 O75604 1/20 0.45
TP53 P04637 1/20 0.45
GAA P10253 1/20 0.45
CASP1 P29466 1/20 0.45
HTT P42858 1/20 0.45
CASP7 P55210 1/20 0.45
KMT2A Q03164 1/20 0.45
ATM Q13315 1/20 0.45
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
PKM P14618 1/20 0.38
GPR55 Q9Y2T6 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13862935 0.87 ALDH1A1 (0.42) MAPTALDH1A1KDM4EPOLBMEN1
SCHEMBL10158281 0.81 MAPT (0.50) CSNK2A1MAPTALDH1A1KDM4EPOLB
SCHEMBL11868776 0.75 MCHR1 (0.49) MAPTALDH1A1KDM4EPOLBMEN1
SCHEMBL7928280 0.73 MCHR1 (0.58) CSNK2A1MAPTALDH1A1KDM4EPOLB
SCHEMBL22787328 0.72 MAPT (0.44) MAPTALDH1A1KDM4EPOLBMEN1
SCHEMBL3784534 0.71 MCHR1 (0.49) CSNK2A1MAPTALDH1A1KDM4EPOLB
SCHEMBL9410520 0.71 CLCN2 (0.38) CSNK2A1ALDH1A1POLBHTTL3MBTL1
SCHEMBL31569145 0.71 CTRC (0.38) MAPTALDH1A1KDM4EPOLBMEN1
SCHEMBL7849660 0.70 IKBKB (0.46) CSNK2A1MAPTALDH1A1KDM4EPOLB
SCHEMBL11794509 0.69 HSD17B10 (0.46) MAPTALDH1A1KDM4EPOLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2220076-B1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION BOEHRINGER INGELHEIM INT (DE) 2012-01-18 EP disclosed