SCHEMBL10167500

SCHEMBL10167500

CCN(C(=O)C1CC1)C1=NS(=O)(=O)c2cccc(Cl)c21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.37
HPGD P15428 2/20 0.34
GHSR Q92847 1/20 0.34
TP53 P04637 2/20 0.34
RET P07949 1/20 0.34
GRK5 P34947 1/20 0.34
TYRO3 Q06418 1/20 0.34
DYRK1B Q9Y463 1/20 0.34
MAPT P10636 2/20 0.34
KDM4E B2RXH2 2/20 0.34
GAA P10253 2/20 0.34
NPSR1 Q6W5P4 1/20 0.34
KCNA3 P22001 4/20 0.33
CNR2 P34972 1/20 0.33
KCNA5 P22460 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
SLC6A3 Q01959 1/20 0.32
LMNA P02545 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10167477 0.88 TP53 (0.35) HTTHPGDGHSRTP53RET
SCHEMBL10167480 0.83 TP53 (0.37) HTTHPGDTP53RETGRK5
SCHEMBL10167479 0.82 TP53 (0.41) HTTHPGDTP53MAPTKDM4E
SCHEMBL13903579 0.79 HTT (0.43) HTTHPGDGHSRRETGRK5
SCHEMBL13903587 0.78 KCNA3 (0.38) HTTHPGDGHSRRETGRK5
SCHEMBL13903831 0.76 PKM (0.37) HTTHPGDRETGRK5TYRO3
SCHEMBL13903622 0.74 RET (0.38) HTTHPGDRETGRK5TYRO3
SCHEMBL13903578 0.74 RET (0.40) HTTHPGDRETGRK5TYRO3
SCHEMBL4390046 0.74 MAPT (0.39) HTTHPGDMAPTKDM4EGAA
SCHEMBL10167471 0.74 LMNA (0.35) HTTHPGDTP53RETGRK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8119568-B2 3-amino-1,2-benzisothiazole compounds for combating animal pest II BASF SE (DE) 2012-02-21 US disclosed
US-8119568-B2 3-amino-1,2-benzisothiazole compounds for combating animal pest II BASF SE (DE) 2012-02-21 US disclosed
US-20100009848-A1 3-Amino-1,2-Benzisothiazole Compounds for Combating Animal Pest II BASF SE (DE) 2010-01-14 US disclosed
US-20100009848-A1 3-Amino-1,2-Benzisothiazole Compounds for Combating Animal Pest II BASF SE (DE) 2010-01-14 US disclosed
WO-2008090048-A2 3-AMINO-1,2-BENZISOTHIAZOLE COMPOUNDS FOR COMBATING ANIMAL PEST II BASF SE (DE) 2008-07-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100009848-A1 3-Amino-1,2-Benzisothiazole Compounds for Combating Animal Pest II BPNT1, BCAT1, TGFBR1 HTT 2470/4885HPGD 4749/4885GHSR 279/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.