SCHEMBL10175445

SCHEMBL10175445

Cn1c(-c2cncc3ccccc23)nc2ccc(F)c(F)c21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 14/20 1.00
CYP11B1 P15538 11/20 0.42
ERN1 O75460 1/20 0.42
PRKCZ Q05513 1/20 0.38
CYP17A1 P05093 2/20 0.37
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2B6 P20813 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL460533 0.83 CYP11B2 (0.71) CYP11B2CYP11B1ERN1CNR1CNR2
SCHEMBL17896768 0.82 CYP11B2 (0.69) CYP11B2CYP11B1ERN1PRKCZCYP17A1
SCHEMBL17896708 0.81 CYP11B2 (0.68) CYP11B2CYP11B1CYP3A4
SCHEMBL17883780 0.81 CYP11B2 (0.68) CYP11B2CYP11B1ERN1PRKCZCYP17A1
SCHEMBL460601 0.81 CYP11B2 (0.67) CYP11B2CYP11B1ERN1PRKCZCNR1
SCHEMBL10175463 0.80 CYP11B2 (0.67) CYP11B2CYP11B1CYP3A4
SCHEMBL463351 0.80 CYP11B2 (0.67) CYP11B2CYP11B1CYP17A1
SCHEMBL10175451 0.77 CYP11B2 (0.63) CYP11B2CYP11B1
SCHEMBL17896706 0.76 CYP11B2 (0.61) CYP11B2CYP11B1
SCHEMBL17897047 0.76 CYP11B2 (0.61) CYP11B2CYP11B1CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed