SCHEMBL10175463

SCHEMBL10175463

Cc1cncc(-c2nc3ccc(F)c(F)c3n2C)c1C

nearest known ligand 0.67

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 7/20 0.67
CYP11B1 P15538 6/20 0.47
CYP3A4 P08684 1/20 0.37
SSTR5 P35346 1/20 0.32
PDE10A Q9Y233 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17896708 0.90 CYP11B2 (0.68) CYP11B2CYP11B1CYP3A4SSTR5
SCHEMBL17897047 0.84 CYP11B2 (0.61) CYP11B2CYP11B1CYP3A4PDE10A
SCHEMBL463351 0.83 CYP11B2 (0.67) CYP11B2CYP11B1PDE10A
SCHEMBL10175451 0.83 CYP11B2 (0.63) CYP11B2CYP11B1PDE10A
SCHEMBL460501 0.83 CYP11B2 (0.63) CYP11B2CYP11B1CYP3A4
SCHEMBL10175445 0.80 CYP11B2 (1.00) CYP11B2CYP11B1CYP3A4
SCHEMBL17896706 0.76 CYP11B2 (0.61) CYP11B2CYP11B1PDE10A
SCHEMBL10175449 0.76 CYP11B2 (0.60) CYP11B2CYP11B1PDE10A
SCHEMBL10176205 0.75 CYP11B2 (0.56) CYP11B2CYP11B1
SCHEMBL10175459 0.75 CYP11B2 (0.56) CYP11B2CYP11B1PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed