SCHEMBL10175456

SCHEMBL10175456

Cn1c(-c2ccncc2)nc2cc(C#N)ccc21

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.57
KMT2A Q03164 1/20 0.57
CYP11B2 P19099 3/20 0.48
ATM Q13315 1/20 0.48
PKN1 Q16512 1/20 0.45
PKN2 Q16513 1/20 0.45
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA9 Q16790 1/20 0.44
KDM4E B2RXH2 3/20 0.43
ALDH1A1 P00352 3/20 0.43
GAA P10253 2/20 0.43
GLA P06280 1/20 0.43
NPC1 O15118 2/20 0.41
TP53 P04637 2/20 0.41
RAB9A P51151 2/20 0.41
HSD17B10 Q99714 2/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17897060 0.89 MEN1 (0.57) MEN1KMT2ACYP11B2ATMPKN1
SCHEMBL13749911 0.87 ATM (0.52) MEN1KMT2ACYP11B2ATMCA12
SCHEMBL4243953 0.84 CYP11B2 (0.69) CYP11B2ATMCYP11B1NAMPT
SCHEMBL10175348 0.82 CYP11B2 (0.48) MEN1KMT2ACYP11B2ATMCA12
SCHEMBL10249140 0.80 MEN1 (0.66) MEN1KMT2AATMCA12CA1
SCHEMBL17896641 0.80 CYP11B2 (0.47) CYP11B2ATMKDM4EALDH1A1GAA
SCHEMBL10175342 0.80 CYP11B2 (0.46) CYP11B2ATMCA12CA1CA2
SCHEMBL12217711 0.79 KDM4E (0.56) MEN1KMT2ACA12CA1CA2
SCHEMBL10953589 0.79 KDM4E (0.50) MEN1KMT2ACYP11B2KDM4EALDH1A1
SCHEMBL17896642 0.78 ALOX5AP (0.46) CYP11B2CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed