SCHEMBL10187301

SCHEMBL10187301

Nc1nc(OCC2CC2)ccc1Br

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EP300 Q09472 5/20 0.41
CNR2 P34972 2/20 0.38
KDM1A O60341 2/20 0.38
CCNA2 P20248 2/20 0.37
CDK2 P24941 2/20 0.37
CCNA1 P78396 2/20 0.37
LRRK2 Q5S007 1/20 0.36
MCHR1 Q99705 3/20 0.35
CDK1 P06493 1/20 0.35
PARP15 Q460N3 1/20 0.35
PARP10 Q53GL7 1/20 0.35
PARP2 Q9UGN5 1/20 0.35
DHFR P00374 1/20 0.35
DCPS Q96C86 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19963006 0.80 EP300 (0.41) EP300CNR2KDM1ACCNA2CDK2
SCHEMBL9966863 0.78 KDM1A (0.40) EP300CNR2KDM1ACCNA2CDK2
SCHEMBL10187309 0.75 ALDH1A1 (0.39) DHFR
SCHEMBL20772826 0.74 CCNA2 (0.41) EP300CNR2KDM1ACCNA2CDK2
SCHEMBL10485526 0.74 CCNA2 (0.44) EP300CNR2CCNA2CDK2CCNA1
SCHEMBL5280 0.72 HTR7 (0.50) EP300CNR2KDM1ACCNA2CDK2
SCHEMBL2728360 0.72 MCHR1 (0.50) EP300CNR2KDM1ACCNA2CDK2
SCHEMBL22834474 0.72 NUDT1 (0.53) EP300CCNA2CDK2CCNA1LRRK2
SCHEMBL30350618 0.72 HTR7 (0.50) EP300CNR2KDM1ACCNA2CDK2
SCHEMBL20772824 0.72 CDK2 (0.39) EP300CNR2KDM1ACCNA2CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012001107-A1 PIPERIDINE DERIVATIVES AND THEIR USE FOR THE TREATMENT OF METABOLIC DISORDERS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-01-05 WO disclosed