SCHEMBL902450

SCHEMBL902450

COC(=O)C[C@H]1CC[C@H](c2ccc(-c3ccc(-c4nc5ccc(C(=O)OC)cc5[nH]4)cc3)cc2)CC1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 8/20 0.60
SOAT1 P35610 2/20 0.60
MMP2 P08253 1/20 0.53
MMP9 P14780 1/20 0.53
MMP8 P22894 1/20 0.53
MMP13 P45452 1/20 0.53
RHEB Q15382 1/20 0.49
KDM4E B2RXH2 1/20 0.49
NPC1 O15118 1/20 0.49
ALDH1A1 P00352 1/20 0.49
LMNA P02545 1/20 0.49
PKM P14618 1/20 0.49
HPGD P15428 1/20 0.49
NFKB1 P19838 1/20 0.49
RAB9A P51151 1/20 0.49
NFKB2 Q00653 1/20 0.49
RELA Q04206 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
SIRT2 Q8IXJ6 3/20 0.48
SIRT1 Q96EB6 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10189188 0.82 DGAT1 (0.56) DGAT1SOAT1RHEBCHEK2
SCHEMBL20982471 0.80 MMP2 (0.78) MMP2MMP9MMP8MMP13RHEB
SCHEMBL10189104 0.80 DGAT1 (0.52) DGAT1SOAT1RHEB
SCHEMBL10189200 0.79 DGAT1 (0.71) DGAT1SOAT1
SCHEMBL14984444 0.78 ALDH1A1 (0.48) DGAT1KDM4ENPC1ALDH1A1LMNA
SCHEMBL901818 0.77 DGAT1 (0.49) DGAT1SOAT1
SCHEMBL19763371 0.76 CHEK2 (0.72) MMP2MMP9MMP8MMP13RHEB
SCHEMBL902547 0.75 DGAT1 (0.78) DGAT1SOAT1
SCHEMBL19747752 0.75 MMP2 (0.70) MMP2MMP9MMP8MMP13RHEB
SCHEMBL2617479 0.74 KDM4E (0.71) MMP2MMP9MMP8MMP13RHEB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012044567-A2 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed