SCHEMBL902206

SCHEMBL902206

Clc1ccc2nc(-c3ccc(-c4ccc(C5CCCCC5)cc4)cn3)[nH]c2c1

nearest known ligand 0.61

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 13/20 0.61
SOAT1 P35610 5/20 0.55
KCNH2 Q12809 10/20 0.53
NPC1 O15118 1/20 0.53
METAP2 P50579 2/20 0.50
METAP1 P53582 2/20 0.50
CBFB Q13951 1/20 0.50
ADORA3 P0DMS8 1/20 0.48
RIPK1 Q13546 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10189200 0.80 DGAT1 (0.71) DGAT1SOAT1KCNH2
SCHEMBL900860 0.80 DGAT1 (0.63) DGAT1SOAT1KCNH2
SCHEMBL10189573 0.79 DGAT1 (0.55) DGAT1SOAT1NPC1RIPK1
SCHEMBL10189566 0.76 DGAT1 (0.77) DGAT1SOAT1KCNH2
SCHEMBL902557 0.76 DGAT1 (0.86) DGAT1SOAT1KCNH2
SCHEMBL4181947 0.75 NPC1 (0.59) DGAT1SOAT1KCNH2NPC1METAP2
SCHEMBL4183736 0.74 CBFB (0.81) NPC1METAP2METAP1CBFBADORA3
SCHEMBL4182090 0.73 METAP2 (0.62) DGAT1SOAT1KCNH2NPC1METAP2
SCHEMBL10189208 0.72 S1PR1 (0.42) DGAT1NPC1CBFB
SCHEMBL902210 0.71 PKN1 (0.60) DGAT1SOAT1KCNH2METAP2METAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012044567-A2 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed