SCHEMBL10195458

SCHEMBL10195458

N=C(c1cn(-c2ccc(C(=O)N3CCOCC3)cc2)nn1)c1cc(C2=CCN(Cc3ccccc3)CC2)ccc1N

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.42
DRD4 P21917 2/20 0.42
DRD3 P35462 2/20 0.42
ALDH1A1 P00352 5/20 0.38
PKM P14618 1/20 0.38
HDAC4 P56524 1/20 0.38
NAMPT P43490 1/20 0.38
HTR1A P08908 1/20 0.38
GAA P10253 2/20 0.37
IDO1 P14902 1/20 0.37
TDO2 P48775 1/20 0.37
HPGD P15428 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
ESRRA P11474 1/20 0.35
TSHR P16473 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17850414 0.78 HPGD (0.40) ALDH1A1GAAIDO1TDO2HPGD
SCHEMBL10194984 0.78 CDC7 (0.44) DRD2DRD4DRD3ALDH1A1PKM
SCHEMBL10194916 0.74 IDO1 (0.42) ALDH1A1PKMGAAIDO1TDO2
SCHEMBL17850419 0.72 WDR5 (0.37) ALDH1A1HPGDKMT2A
SCHEMBL10194732 0.69 ESRRA (0.44) ALDH1A1GAAESRRATSHRL3MBTL1
SCHEMBL10195780 0.68 ESRRA (0.44) ALDH1A1ESRRATSHRL3MBTL1HTT
SCHEMBL10195446 0.67 PIK3CA (0.42) HPGDSMN1; SMN2MEN1KMT2AESRRA
SCHEMBL17850412 0.66 ESRRA (0.48) SMN1; SMN2ESRRA
SCHEMBL4030523 0.65 HDAC4 (0.61) DRD2DRD4DRD3HDAC4NAMPT
SCHEMBL2396123 0.64 HDAC4 (0.58) DRD2DRD4DRD3ALDH1A1HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012084704-A1 INDAZOLYL TRIAZOLE DERIVATIVES AS IRAK INHIBITORS MERCK SERONO S.A. (CH) 2012-06-28 WO disclosed