SCHEMBL17850419

SCHEMBL17850419

N=C(c1cn(-c2ccc(C(=O)N3CCOCC3)cc2)nn1)c1cc(C2CCN(CCF)CC2)ccc1N

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
WDR5 P61964 4/20 0.37
KMT2A Q03164 2/20 0.35
HRH3 Q9Y5N1 3/20 0.34
HTR2B P41595 1/20 0.34
KDM1A O60341 2/20 0.34
HDAC6 Q9UBN7 2/20 0.34
JAK2 O60674 1/20 0.33
HPGDS O60760 1/20 0.33
HPGD P15428 2/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPK14 Q16539 1/20 0.33
APC P25054 2/20 0.33
BMPR1B O00238 1/20 0.33
BMPR1A P36894 1/20 0.33
TGFBR1 P36897 1/20 0.33
ACVRL1 P37023 1/20 0.33
ACVR1 Q04771 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17850414 0.80 HPGD (0.40) WDR5JAK2HPGDALDH1A1
SCHEMBL10194739 0.77 FLT3 (0.43) HTR2BJAK2MAPK14
SCHEMBL10194916 0.73 IDO1 (0.42) WDR5KMT2AHPGDALDH1A1
SCHEMBL10195458 0.72 DRD2 (0.42) KMT2AHPGDALDH1A1
SCHEMBL10195780 0.69 ESRRA (0.44) WDR5ALDH1A1
SCHEMBL10196924 0.68 L3MBTL3 (0.43) HRH3HPGDALDH1A1
SCHEMBL10195446 0.68 PIK3CA (0.42) WDR5KMT2AHPGD
SCHEMBL10195439 0.68 PHGDH (0.35) KMT2AHTR2BJAK2HPGDALDH1A1
SCHEMBL10194732 0.67 ESRRA (0.44) WDR5ALDH1A1
SCHEMBL17850412 0.67 ESRRA (0.48) WDR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2655357-B1 INDAZOLYL TRIAZOLE DERIVATIVES AS IRAK INHIBITORS MERCK SERONO SA (CH) 2016-06-22 EP disclosed