SCHEMBL17850414

SCHEMBL17850414

N=C(c1cn(-c2ccc(C(=O)N3CCOCC3)cc2)nn1)c1cc(CO)ccc1N

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HPGD P15428 6/20 0.40
SMN1; SMN2 Q16637 5/20 0.40
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.40
MAPT P10636 1/20 0.40
HTT P42858 1/20 0.40
IDO1 P14902 1/20 0.39
TDO2 P48775 1/20 0.39
WDR5 P61964 1/20 0.39
GAA P10253 2/20 0.38
ESRRA P11474 1/20 0.37
PHGDH O43175 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
JAK2 O60674 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C19 P33261 1/20 0.37
MAPK10 P53779 1/20 0.36
LRRK2 Q5S007 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10194916 0.85 IDO1 (0.42) HPGDSMN1; SMN2ALDH1A1IDO1TDO2
SCHEMBL10195752 0.81 GPR119 (0.40) HPGDSMN1; SMN2ALDH1A1KDM4EMAPT
SCHEMBL17850419 0.80 WDR5 (0.37) HPGDALDH1A1WDR5JAK2
SCHEMBL10195458 0.78 DRD2 (0.42) HPGDSMN1; SMN2ALDH1A1HTTIDO1
SCHEMBL10195780 0.73 ESRRA (0.44) ALDH1A1MAPTHTTWDR5ESRRA
SCHEMBL10194732 0.73 ESRRA (0.44) ALDH1A1KDM4EMAPTHTTWDR5
SCHEMBL10195446 0.73 PIK3CA (0.42) HPGDSMN1; SMN2WDR5ESRRANPC1
SCHEMBL10194789 0.71 MAPK10 (0.47) HPGDSMN1; SMN2ALDH1A1KDM4EMAPT
SCHEMBL10194698 0.71 MAPK10 (0.49) HPGDSMN1; SMN2ALDH1A1KDM4EMAPT
SCHEMBL17850412 0.71 ESRRA (0.48) SMN1; SMN2WDR5ESRRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2655357-B1 INDAZOLYL TRIAZOLE DERIVATIVES AS IRAK INHIBITORS MERCK SERONO SA (CH) 2016-06-22 EP disclosed