SCHEMBL10202053

SCHEMBL10202053

CS(=O)(=O)NC(=O)c1ccc(CBr)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 3/20 0.50
P4HTM Q9NXG6 2/20 0.47
PTPN1 P18031 1/20 0.47
CES2 O00748 1/20 0.46
CES1 P23141 1/20 0.46
KDM4E B2RXH2 2/20 0.45
POLB P06746 1/20 0.45
TSHR P16473 1/20 0.45
RECQL P46063 1/20 0.45
SCN3A Q9NY46 1/20 0.45
KMT2A Q03164 1/20 0.45
HDAC6 Q9UBN7 4/20 0.44
HDAC8 Q9BY41 2/20 0.44
HDAC1 Q13547 2/20 0.42
MAP4K4 O95819 1/20 0.42
PLK1 P53350 1/20 0.42
HDAC3 O15379 1/20 0.42
NCOR2 Q9Y618 1/20 0.42
EPHX2 P34913 1/20 0.41
NR1H4 Q96RI1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8442436 0.86 SCN9A (0.48) SCN9AP4HTMPTPN1KDM4EPOLB
SCHEMBL7973340 0.84 PLK1 (0.61) SCN9AP4HTMPTPN1KDM4EPOLB
SCHEMBL13141179 0.82 HDAC6 (0.65) SCN9AP4HTMPTPN1KDM4EPOLB
SCHEMBL7118965 0.79 ALDH1A1 (0.58) SCN9AP4HTMPTPN1CES2CES1
SCHEMBL8337823 0.79 THRA (0.50) SCN9AP4HTMPTPN1KDM4EPOLB
SCHEMBL279954 0.77 HDAC1 (0.63) SCN9AP4HTMPTPN1CES2CES1
SCHEMBL17629544 0.77 PLK1 (0.68) CES2CES1POLBTSHRKMT2A
SCHEMBL10235812 0.76 MCL1 (0.49) SCN9A
SCHEMBL7990845 0.76 FLT1 (0.65) SCN9AP4HTMKDM4EPOLBMAP4K4
SCHEMBL9913954 0.76 KMT2A (0.54) SCN9AP4HTMPTPN1KMT2AEPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117120416-A Small molecule compound with substituted phenyl spiro [ indoline-3, 3' -pyrrolidine ] structure 中国科学院上海药物研究所 2023-11-24 CN disclosed
CN-115215872-A Small molecule compound with substituted phenyl spiro [ indoline-3, 3' -pyrrolidine ] structure 中国科学院上海药物研究所 2022-10-21 CN disclosed
US-9096500-B2 Acyl sulfonamide compounds PFIZER LIMITED (GB) 2015-08-04 US disclosed
US-9096500-B2 Acyl sulfonamide compounds PFIZER LIMITED (GB) 2015-08-04 US disclosed
US-9096500-B2 Acyl sulfonamide compounds PFIZER LIMITED (GB) 2015-08-04 US disclosed
EP-2593428-B1 N-SULFONYLBENZAMIDES AS INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS PFIZER LTD (GB) 2014-11-19 EP disclosed
EP-2593428-B1 N-SULFONYLBENZAMIDES AS INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS PFIZER LTD (GB) 2014-11-19 EP disclosed
US-20130109701-A1 Chemical Compounds PFIZER LIMITED (GB) 2013-05-02 US disclosed
US-20130109701-A1 Chemical Compounds PFIZER LIMITED (GB) 2013-05-02 US disclosed
US-20130109701-A1 Chemical Compounds PFIZER LIMITED (GB) 2013-05-02 US disclosed
WO-2012007868-A2 CHEMICAL COMPOUNDS PFIZER LIMITED (GB) 2012-01-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130109701-A1 Chemical Compounds SCN1A, SCN1B, SCN7A SCN9A 16/4885P4HTM 3138/4885PTPN1 419/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.