SCHEMBL7118965

SCHEMBL7118965

CS(=O)(=O)NC(=O)c1ccc(Br)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.58
SCN9A Q15858 1/20 0.54
OGG1 O15527 1/20 0.53
P4HTM Q9NXG6 2/20 0.51
PTGS1 P23219 2/20 0.51
PTGS2 P35354 2/20 0.51
HDAC1 Q13547 2/20 0.47
HDAC2 Q92769 2/20 0.47
HDAC3 O15379 1/20 0.47
PTPN1 P18031 1/20 0.47
CES2 O00748 1/20 0.46
CES1 P23141 1/20 0.46
POLB P06746 1/20 0.46
CTDSP1 Q9GZU7 1/20 0.46
CA12 O43570 1/20 0.46
MMP2 P08253 1/20 0.46
CA14 Q9ULX7 1/20 0.46
HDAC6 Q9UBN7 2/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6608459 0.94 SCN9A (0.62) ALDH1A1SCN9AOGG1P4HTMPTGS1
SCHEMBL279954 0.82 HDAC1 (0.63) ALDH1A1SCN9AP4HTMPTGS2HDAC1
SCHEMBL7990884 0.81 OGG1 (0.55) ALDH1A1OGG1PTGS1PTGS2HDAC1
SCHEMBL7987812 0.80 SCN9A (0.55) SCN9AP4HTMPTGS1PTGS2PTPN1
SCHEMBL22097521 0.80 SCN9A (0.54) SCN9AP4HTMHDAC1HDAC2PTPN1
SCHEMBL7990845 0.80 FLT1 (0.65) ALDH1A1SCN9AP4HTMPTGS1PTGS2
SCHEMBL3374779 0.80 SCN9A (0.54) ALDH1A1SCN9AP4HTMPTPN1CA12
SCHEMBL9913954 0.80 KMT2A (0.54) ALDH1A1SCN9AP4HTMPTPN1CA2
SCHEMBL1647742 0.80 LMNA (0.54) ALDH1A1SCN9AP4HTMPTPN1POLB
SCHEMBL10202053 0.79 SCN9A (0.50) SCN9AP4HTMHDAC1HDAC3PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0793656-B1 NOVEL BENZYL PYRIMIDINES BASILEA PHARMACEUTICA AG (CH) 2003-03-26 EP disclosed
US-6331628-B1 REACTING A SUBSTITUTED HALOBENZENE WITH POTASSIUM, SODIUM AND/OR ZINC CYANIDE IN THE PRESENCE OF A METALLIC CATALYST NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2001-12-18 US disclosed
US-5763450-A BACTERICIDES; TREATMENT OF INFECTIOUS DISEASES HOFFMANN-LA ROCHE INC. (US) 1998-06-09 US disclosed
EP-0793656-A1 NOVEL BENZYL PYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 1997-09-10 EP disclosed
WO-1996016046-A2 NOVEL BENZYL PYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 1996-05-30 WO disclosed