SCHEMBL1020544

SCHEMBL1020544

CNc1cccc(-n2cncn2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.49
BRD4 O60885 1/20 0.45
CREBBP Q92793 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
S1PR1 P21453 1/20 0.41
CHRNA7 P36544 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2D6 P10635 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
CYP3A4 P08684 1/20 0.37
GRK6 P43250 1/20 0.37
MAPK10 P53779 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5252164 0.83 HDAC1 (0.45) CYP2A6BRD4CREBBPSMN1; SMN2KDM4E
SCHEMBL11926858 0.82 CYP2A6 (0.62) CYP2A6BRD4CREBBPSMN1; SMN2KDM4E
SCHEMBL14076589 0.79 SMN1; SMN2 (0.55) CYP2A6BRD4CREBBPSMN1; SMN2KDM4E
SCHEMBL4457861 0.78 S1PR1 (0.47) CYP2A6BRD4CREBBPSMN1; SMN2KDM4E
SCHEMBL9454459 0.77 CYP2A6 (0.53) CYP2A6SMN1; SMN2KDM4EALDH1A1CHRNA7
SCHEMBL18974765 0.77 KMT2A (0.47) CYP2A6BRD4CREBBPSMN1; SMN2KDM4E
SCHEMBL23289039 0.76 CYP1A2 (0.42) CYP2A6SMN1; SMN2KDM4EALDH1A1CYP1A2
SCHEMBL10154296 0.76 PRMT6 (0.50) CYP2A6SMN1; SMN2KDM4EALDH1A1CHRNA7
SCHEMBL5328745 0.75 GRK6 (0.47) CYP2A6BRD4CREBBPSMN1; SMN2KDM4E
SCHEMBL4948621 0.75 LMNA (0.47) SMN1; SMN2KDM4EALDH1A1MAPK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114206870-A Tricyclic AKR1C3 dependent KARS inhibitors 诺华股份有限公司 2022-03-18 CN disclosed
US-20190019964-A1 ORGANOMETALLIC COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME SAMSUNG DISPLAY CO., LTD. (KR) 2019-01-17 US disclosed
US-7960556-B2 Thiadiazole derivatives for the treatment of neuro-degenerative diseases NV REMYND (BE) 2011-06-14 US disclosed
EP-2094677-B1 THIADIAZOLE DERIVATIVES FOR THE TREATMENT OF NEURO-DEGENERATIVE DISEASES REMYND NV (BE) 2011-01-12 EP disclosed
US-20100144709-A1 THIADIAZOLE DERIVATIVES FOR THE TREATMENT OF NEURO-DEGENERATIVE DISEASES NV REMYND (BE) 2010-06-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190019964-A1 ORGANOMETALLIC COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME LEF1, OCIAD1, POU2F1 CYP2A6 2757/4885BRD4 3758/4885CREBBP 2461/4885
US-20100144709-A1 THIADIAZOLE DERIVATIVES FOR THE TREATMENT OF NEURO-DEGENERATIVE DISEASES SNCA, PARK7, PRNP CYP2A6 4301/4885BRD4 224/4885CREBBP 260/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.