SCHEMBL102179

SCHEMBL102179

CCOc1cc(NC(=O)CCCc2ccc(-c3ccccc3)c(NC(=O)O)c2)ccc1CO[Si](C)(C)C(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.42
RAB9A P51151 3/20 0.42
MAPT P10636 4/20 0.40
BRD4 O60885 1/20 0.39
POLB P06746 1/20 0.38
CNR2 P34972 1/20 0.37
THRB P10828 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP3A4 P08684 1/20 0.36
TSHR P16473 1/20 0.36
MAPKAPK2 P49137 1/20 0.36
KMT2A Q03164 1/20 0.36
NR2E1 Q9Y466 1/20 0.36
ITGB1 P05556 1/20 0.36
ITGA4 P13612 1/20 0.36
TRPV1 Q8NER1 1/20 0.36
NFKB1 P19838 1/20 0.35
NFKB2 Q00653 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL99375 0.92 NPC1 (0.49) NPC1RAB9AMAPTPOLBSMN1; SMN2
SCHEMBL99141 0.91 NPC1 (0.48) NPC1RAB9AMAPTPOLBCNR2
SCHEMBL99117 0.89 CHEK1 (0.38) NPC1RAB9AMAPTPOLBSMN1; SMN2
SCHEMBL99071 0.88 RAB9A (0.43) NPC1RAB9ASMN1; SMN2MEN1TSHR
SCHEMBL100167 0.88 SMN1; SMN2 (0.43) NPC1RAB9AMAPTPOLBCNR2
SCHEMBL102612 0.87 NPC1 (0.48) NPC1RAB9AMAPTBRD4POLB
SCHEMBL663672 0.86 CHRM3 (0.44)
SCHEMBL102843 0.86 HCAR2 (0.42) NPC1RAB9AMAPTPOLBSMN1; SMN2
SCHEMBL98208 0.85 HCAR2 (0.41) NPC1RAB9AMAPTPOLBCNR2
SCHEMBL100524 0.84 RORC (0.43) NPC1RAB9AMAPTSMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426121-A1 QUATERNARY AMMONIUM SALT COMPOUND Teijin Pharma Limited (JP) 2012-03-07 EP claimed