SCHEMBL99375

SCHEMBL99375

COc1cc(NC(=O)CCCc2ccc(-c3ccccc3)c(NC(=O)O)c2)ccc1CO[Si](C)(C)C(C)(C)C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
HPGD P15428 2/20 0.41
POLB P06746 2/20 0.40
MAPT P10636 2/20 0.40
HDAC1 Q13547 2/20 0.38
HDAC2 Q92769 2/20 0.38
KMT2A Q03164 3/20 0.38
IMPDH2 P12268 2/20 0.38
MEN1 O00255 2/20 0.38
TSHR P16473 2/20 0.38
AAK1 Q2M2I8 1/20 0.38
HDAC3 O15379 1/20 0.38
IMPDH1 P20839 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC10 Q969S8 1/20 0.38
HDAC11 Q96DB2 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL99141 0.98 NPC1 (0.48) NPC1RAB9AHPGDPOLBMAPT
SCHEMBL99071 0.96 RAB9A (0.43) NPC1RAB9AHDAC1HDAC2KMT2A
SCHEMBL102179 0.92 NPC1 (0.42) NPC1RAB9APOLBMAPTKMT2A
SCHEMBL102843 0.89 HCAR2 (0.42) NPC1RAB9APOLBMAPTHDAC1
SCHEMBL100167 0.89 SMN1; SMN2 (0.43) NPC1RAB9APOLBMAPTHDAC1
SCHEMBL99659 0.88 POLB (0.40) NPC1RAB9AHPGDPOLBMAPT
SCHEMBL97653 0.88 CHEK1 (0.42) NPC1RAB9AHPGDPOLBMAPT
SCHEMBL98208 0.87 HCAR2 (0.41) NPC1RAB9AHPGDPOLBMAPT
SCHEMBL99703 0.86 NPC1 (0.58) NPC1RAB9AHPGDPOLBMAPT
SCHEMBL663959 0.86 CHRM3 (0.46) NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426121-A1 QUATERNARY AMMONIUM SALT COMPOUND Teijin Pharma Limited (JP) 2012-03-07 EP claimed