SCHEMBL99071

SCHEMBL99071

COc1cc(NC(=O)CCc2ccc(-c3ccccc3)c(NC(=O)O)c2)ccc1CO[Si](C)(C)C(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.43
NPC1 O15118 1/20 0.43
KMT2A Q03164 2/20 0.42
TSHR P16473 1/20 0.42
HDAC1 Q13547 5/20 0.42
HDAC2 Q92769 5/20 0.42
LTB4R Q15722 1/20 0.41
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
MEN1 O00255 1/20 0.39
IMPDH2 P12268 2/20 0.39
AAK1 Q2M2I8 1/20 0.39
GAA P10253 1/20 0.38
PKM P14618 1/20 0.38
HCAR2 Q8TDS4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL99375 0.96 NPC1 (0.49) RAB9ANPC1KMT2ATSHRHDAC1
SCHEMBL99141 0.94 NPC1 (0.48) RAB9ANPC1KMT2ATSHRHDAC1
SCHEMBL102843 0.93 HCAR2 (0.42) RAB9ANPC1KMT2ATSHRHDAC1
SCHEMBL101812 0.89 PTGDR2 (0.42) RAB9ANPC1HDAC1HDAC2HCAR2
SCHEMBL100524 0.89 RORC (0.43) RAB9ANPC1KMT2ATSHRHDAC1
SCHEMBL102179 0.88 NPC1 (0.42) RAB9ANPC1KMT2ATSHRLMNA
SCHEMBL99813 0.88 HCAR2 (0.44) RAB9AHDAC1HDAC2HCAR2
SCHEMBL100322 0.87 HPGD (0.44) RAB9ANPC1KMT2ATSHRHDAC1
SCHEMBL98766 0.86 LTB4R (0.52) KMT2ATSHRLTB4RSMN1; SMN2MEN1
SCHEMBL99091 0.86 RAB9A (0.51) RAB9ANPC1KMT2ATSHRHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426121-A1 QUATERNARY AMMONIUM SALT COMPOUND Teijin Pharma Limited (JP) 2012-03-07 EP claimed