SCHEMBL1025531

SCHEMBL1025531

NC(=O)c1ccc2c(c1)CCNC2OC1CCCCO1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 7/20 0.36
HTR1B P28222 3/20 0.36
DRD2 P14416 5/20 0.36
HTR2A P28223 3/20 0.36
HTR1A P08908 2/20 0.36
DRD4 P21917 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
MAPKAPK2 P49137 1/20 0.35
NNMT P40261 1/20 0.34
CYP2C9 P11712 1/20 0.34
HPGD P15428 1/20 0.34
AKR1C3 P42330 3/20 0.34
HSD11B1 P28845 1/20 0.34
DRD3 P35462 3/20 0.33
SLC6A4 P31645 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26101504 0.76 NNMT (0.44) HTR1DDRD2HTR2AHTR1ADRD4
SCHEMBL1075684 0.71 DRD3 (0.44) HTR1DHTR1BDRD2MEN1KMT2A
SCHEMBL31511358 0.70 ALDH1A1 (0.40) MEN1KMT2AHPGDHSD11B1
SCHEMBL31511366 0.70 ALDH1A1 (0.40) MEN1KMT2AHPGDHSD11B1
SCHEMBL1026289 0.69 OPRM1 (0.36) MEN1KMT2A
SCHEMBL7389468 0.68 MEN1 (0.42) DRD2MEN1KMT2ADRD3
SCHEMBL20504355 0.68 MAPKAPK2 (0.44) DRD2MEN1KMT2AMAPKAPK2NNMT
SCHEMBL20504221 0.68 PRCP (0.53) DRD2DRD4MEN1KMT2AMAPKAPK2
SCHEMBL26452181 0.68 PARP10 (0.58) MEN1KMT2ACYP2C9HPGD
SCHEMBL1025073 0.66 F2 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2274283-A1 NOVEL N-SUBSTITUTED TETRAHYDROISOQUINOLINE/ISOINDOLINE HYDROXAMIC ACID COMPOUNDS 4SC AG (DE) 2011-01-19 EP disclosed
WO-2009112550-A1 NOVEL N-SUBSTITUTED TETRAHYDROISOQUINOLINE/ISOINDOLINE HYDROXAMIC ACID COMPOUNDS 4SC AG (DE) 2009-09-17 WO disclosed