SCHEMBL10276312

SCHEMBL10276312

CC1=C(c2ccc(C(=O)O)cc2)C=C2NC(c3ccc(C#N)cc3)=CC(=O)N2N1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.39
RARA P10276 1/20 0.36
RARB P10826 1/20 0.36
RARG P13631 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAP4K4 O95819 1/20 0.34
PTPN11 Q06124 1/20 0.34
SIRT5 Q9NXA8 1/20 0.34
NR3C2 P08235 6/20 0.33
RXRA P19793 2/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
SLC22A12 Q96S37 1/20 0.32
MMP2 P08253 1/20 0.32
MMP9 P14780 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10275638 0.78 KCNH2 (0.36) AR
SCHEMBL10276004 0.69 KCNH2 (0.37) AR
SCHEMBL10275809 0.69 NR3C2 (0.39) ARRARARARBRARGALDH1A1
SCHEMBL307426 0.66 MAP4K4 (0.60) ARMAP4K4RXRACA1CA2
Hydrochloric Acid SCHEMBL15939679 0.65 MAP4K4 (0.59) ARMAP4K4RXRACA1CA2
SCHEMBL10275578 0.65 SIRT5 (0.40) ARRARARARBRARGMAP4K4
SCHEMBL23037552 0.65 CA2 (0.59) ARRARBRARGALDH1A1MAP4K4
SCHEMBL216706 0.65 CA2 (0.64) ARRARBRARGALDH1A1MAP4K4
Terephthalic Acid SCHEMBL27298641 0.64 ALDH1A1 (0.68) ARRARBRARGALDH1A1MAP4K4
SCHEMBL10275694 0.63 TDP2 (0.35) ALDH1A1NR3C2CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120178915-A1 PYRIMIDINE DERIVATIVES AND ANALOGS, PREPARATION METHOD AND USE THEREOF XU LIFENG (US) 2012-07-12 US claimed
CN-103554111-A Aromatic heterocyclic pyridine derivatives and analogs, and preparation method and application thereof LIAONING LIFENG SCIENCE AND TECHNOLOGY DEV CO LTD 2014-02-05 CN disclosed
CN-101671336-B Aromatic heterocyclic pyrimidine derivative and analogue, preparation method and application thereof LIAONING LIFENG SCIENCE AND TECHNOLOGY DEV CO LTD 2013-11-13 CN disclosed
US-20120178915-A1 PYRIMIDINE DERIVATIVES AND ANALOGS, PREPARATION METHOD AND USE THEREOF XU LIFENG (US) 2012-07-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120178915-A1 PYRIMIDINE DERIVATIVES AND ANALOGS, PREPARATION METHOD AND USE THEREOF TYMP, TYMS, ADORA3 AR 3221/4885RARA 1915/4885RARB 2365/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.