SCHEMBL1028700

SCHEMBL1028700

O=C(Cc1ccccc1)O[C@H]1CCC[C@@H]1N1C(=O)C=CC1=O

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.43
KMT2A Q03164 3/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
HPGD P15428 2/20 0.42
ALDH1A1 P00352 2/20 0.42
GLA P06280 1/20 0.42
MAPK1 P28482 2/20 0.40
SLC18A3 Q16572 1/20 0.40
MGLL Q99685 2/20 0.39
MAPT P10636 1/20 0.38
PAM P19021 1/20 0.38
EPHX2 P34913 1/20 0.38
OPRM1 P35372 1/20 0.37
OPRK1 P41145 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1024747 0.87 SLC18A3 (0.44) L3MBTL1HPGDALDH1A1SLC18A3MGLL
SCHEMBL1024756 0.81 BCHE (0.53) HPGDALDH1A1
SCHEMBL1029324 0.80 SLC18A3 (0.55) KMT2ASLC18A3MAPT
SCHEMBL1027833 0.79 KMT2A (0.44) KMT2AL3MBTL1ALDH1A1MAPTEPHX2
SCHEMBL1028701 0.79 CHRM2 (0.51) CYP19A1KMT2AHPGDALDH1A1SLC18A3
SCHEMBL1028267 0.78 PSEN1 (0.47) MGLL
SCHEMBL1027406 0.78 PSEN1 (0.47) MGLL
SCHEMBL1028000 0.77 ALDH1A1 (0.44) KMT2AL3MBTL1HPGDALDH1A1GLA
SCHEMBL1028275 0.77 SLC18A3 (0.51) HPGDALDH1A1SLC18A3OPRM1OPRK1
SCHEMBL1027579 0.76 LMNA (0.53) L3MBTL1MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1479669-B1 Optically active maleimide derivatives and polymaleimides for use as chiral adsorbent in chromatography TOSOH CORP (JP) 2011-01-19 EP disclosed
US-7645889-B2 Optically active polymaleimide derivatives and process for their production TOSOH CORPORATION (JP) 2010-01-12 US disclosed
US-20080230482-A1 Optically active polymaleimide derivatives and process for their production TOSOH CORPORATION (JP) 2008-09-25 US disclosed
US-7381742-B2 Optically active polymaleimide derivatives and process for their production TOSOH CORPORATION (JP) 2008-06-03 US disclosed
US-20070131616-A1 Optically active maleimide derivatives, optically active polymaleimide derivatives, process for their production, separating media comprising the optically active polymaleimide derivatives and method of separating optically active compounds using them TOSOH CORPORATION (JP) 2007-06-14 US disclosed
US-7186750-B2 Optically active maleimide derivatives, optically active polymaleimide derivatives, process for their production, separating media comprising the optically active polymaleimide derivatives and method of separating optically active compounds using them TOSOH CORPORATION (JP) 2007-03-06 US disclosed
US-20040235937-A1 Optically active maleimide derivatives, optically active polymaleimide derivatives, process for their production, separating media comprising the optically active polymaleimide derivatives and method of separating optically active compounds using them TOSOH CORPORATION (JP) 2004-11-25 US disclosed
EP-1479669-A1 Optically active maleimide derivatives and polymaleimides for use as chiral adsorbent in chromatography Tosoh Corporation (JP) 2004-11-24 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080230482-A1 Optically active polymaleimide derivatives and process for their production CYBA, COASY, MEP1B CYP19A1 882/4885KMT2A 3220/4885L3MBTL1 4503/4885
US-20040235937-A1 Optically active maleimide derivatives, optically active polymaleimide derivatives, process for their production, separating media comprising the optically active polymaleimide derivatives and method of separating optically active compounds using them MACF1, MEP1B, CYBA CYP19A1 1171/4885KMT2A 2453/4885L3MBTL1 4536/4885
US-20070131616-A1 Optically active maleimide derivatives, optically active polymaleimide derivatives, process for their production, separating media comprising the optically active polymaleimide derivatives and method of separating optically active compounds using them MACF1, MEP1B, ACMSD CYP19A1 1205/4885KMT2A 2367/4885L3MBTL1 4555/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.