SCHEMBL1031357

SCHEMBL1031357

Cc1cn(C)c(OC(=O)NCc2ccc(F)cc2C(F)(F)F)c1-c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 13/20 0.46
NTRK1 P04629 3/20 0.44
EPHX2 P34913 4/20 0.41
PPARG P37231 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1032390 0.85 P2RX7 (0.42) P2RX7NTRK1EPHX2PPARG
SCHEMBL1030468 0.83 P2RX7 (0.48) P2RX7NTRK1EPHX2PPARG
SCHEMBL1032752 0.81 EPHX1 (0.40)
SCHEMBL1032699 0.80 EPHX2 (0.42) P2RX7EPHX2PPARG
SCHEMBL1030010 0.76 MAPK14 (0.50) PPARG
SCHEMBL1031886 0.73 METAP2 (0.37)
SCHEMBL1031826 0.72 PTGER4 (0.43) P2RX7PPARG
SCHEMBL1033134 0.71 P2RX7 (0.43) P2RX7NTRK1EPHX2PPARG
SCHEMBL1032701 0.71 ALDH1A1 (0.44)
SCHEMBL1030941 0.70 TP53 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2035375-B1 1,3-DISUBSTITUTED 4-METHYL-1H-PYRROLE-2-CARBOXAMIDES AND THEIR USE FOR THE MANUFACTURE OF MEDICAMENTS GRUENENTHAL GMBH (DE) 2011-01-19 EP claimed
EP-2035375-B1 1,3-DISUBSTITUTED 4-METHYL-1H-PYRROLE-2-CARBOXAMIDES AND THEIR USE FOR THE MANUFACTURE OF MEDICAMENTS GRUENENTHAL GMBH (DE) 2011-01-19 EP disclosed