SCHEMBL10316671

SCHEMBL10316671

O=C(O)NCc1cccc(-c2nc(-c3cccnc3)no2)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.57
MAPK1 P28482 2/20 0.57
CHRNB2 P17787 4/20 0.56
CHRNA5 P30532 4/20 0.56
CHRNA4 P43681 4/20 0.56
POLB P06746 2/20 0.55
CA9 Q16790 1/20 0.55
TP53 P04637 7/20 0.54
SMN1; SMN2 Q16637 6/20 0.54
NPC1 O15118 4/20 0.54
RAB9A P51151 4/20 0.54
MAPT P10636 3/20 0.54
KDM4E B2RXH2 1/20 0.54
HPGD P15428 1/20 0.54
HSD17B10 Q99714 1/20 0.54
S1PR1 P21453 2/20 0.53
NFKB1 P19838 1/20 0.52
NFKB2 Q00653 1/20 0.52
RELA Q04206 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1423075 0.84 S1PR1 (0.52) ALDH1A1MAPK1CHRNB2CHRNA5CHRNA4
SCHEMBL22501576 0.83 EPHX2 (0.64) SMN1; SMN2NPC1RAB9ACYP1A2CYP3A4
SCHEMBL27767567 0.80 S1PR1 (0.52) ALDH1A1CHRNB2CHRNA5CHRNA4POLB
SCHEMBL4456834 0.80 TP53 (0.62) ALDH1A1CHRNB2CHRNA5CHRNA4POLB
SCHEMBL3715047 0.80 CHRNB2 (0.62) ALDH1A1CHRNB2CHRNA5CHRNA4CA9
SCHEMBL1422372 0.79 KMO (0.67) ALDH1A1CHRNB2CHRNA5CHRNA4POLB
SCHEMBL2273541 0.79 CHRNB2 (0.66) ALDH1A1CHRNB2CHRNA5CHRNA4POLB
Hydrochloric Acid SCHEMBL2278057 0.78 CHRNB2 (0.64) ALDH1A1CHRNB2CHRNA5CHRNA4POLB
SCHEMBL6565112 0.78 L3MBTL1 (0.59) POLBTP53MAPTKMT2ATSHR
SCHEMBL3684765 0.78 TP53 (0.54) ALDH1A1CHRNB2CHRNA5CHRNA4POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2226074-B1 Pharmaceutical compositions and their methods of use ABBVIE INC (US) 2015-11-04 EP claimed
EP-2101763-B1 PHARMACEUTICAL COMPOSITIONS AND THEIR METHODS OF USE ABBOTT LAB (US) 2012-07-18 EP claimed