SCHEMBL1032095

SCHEMBL1032095

Cc1cn(Cc2ccccc2)c(C(=O)NCCc2c[nH]c3ccccc23)c1-c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 4/20 0.56
CCND1 P24385 4/20 0.56
NPC1 O15118 6/20 0.54
RAB9A P51151 6/20 0.54
MEN1 O00255 6/20 0.54
KMT2A Q03164 6/20 0.54
SIRT1 Q96EB6 3/20 0.53
ATM Q13315 1/20 0.52
ACHE P22303 3/20 0.52
CYP1A2 P05177 2/20 0.52
CYP2C19 P33261 2/20 0.52
CYP3A4 P08684 2/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
TSHR P16473 2/20 0.51
LMNA P02545 1/20 0.51
PKM P14618 1/20 0.51
BLM P54132 1/20 0.51
ALDH1A1 P00352 2/20 0.51
MAPT P10636 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1031910 0.85 NPC1 (0.59) CDK4CCND1NPC1RAB9AMEN1
SCHEMBL1030212 0.81 NPC1 (0.61) CDK4CCND1NPC1RAB9AMEN1
SCHEMBL1033446 0.78 NPC1 (0.53) NPC1RAB9AMEN1KMT2ALMNA
SCHEMBL1028192 0.77 HIF1A (0.47) NPC1RAB9AMEN1KMT2ATSHR
SCHEMBL1029726 0.76 PTGS2 (0.52) CDK4CCND1KMT2AACHEMAPT
SCHEMBL1032472 0.75 CDK4 (0.62) CDK4CCND1
SCHEMBL24273323 0.74 SIRT1 (0.62) CDK4CCND1NPC1RAB9AMEN1
SCHEMBL1028264 0.74 CACNA1G (0.47) MEN1KMT2AACHEBCHENPSR1
SCHEMBL1028662 0.73 LMNA (0.48) NPC1RAB9AMEN1KMT2ALMNA
SCHEMBL6394942 0.73 MEN1 (0.76) CDK4CCND1NPC1RAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2035375-B1 1,3-DISUBSTITUTED 4-METHYL-1H-PYRROLE-2-CARBOXAMIDES AND THEIR USE FOR THE MANUFACTURE OF MEDICAMENTS GRUENENTHAL GMBH (DE) 2011-01-19 EP claimed