SCHEMBL1032244

SCHEMBL1032244

COc1ccc(Cn2cc(C)c(-c3ccco3)c2C(=O)NC2CCCc3ccccc32)cc1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.54
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
HTT P42858 1/20 0.47
DHODH Q02127 1/20 0.47
HSD17B10 Q99714 2/20 0.47
RECQL P46063 1/20 0.45
TAS1R3 Q7RTX0 4/20 0.44
TAS1R1 Q7RTX1 4/20 0.44
TAS1R2 Q8TE23 2/20 0.44
CRHBP P24387 1/20 0.44
CRHR2 Q13324 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2637910 0.76 TP53 (0.44) ALDH1A1KMT2A
SCHEMBL1027476 0.76 ALDH1A1 (0.47) ALDH1A1HTTHSD17B10RECQLTAS1R3
SCHEMBL1030586 0.76 ALDH1A1 (0.41) ALDH1A1MEN1KMT2AHTTHSD17B10
SCHEMBL1027735 0.74 ALDH1A1 (0.53) ALDH1A1MEN1KMT2AHTTHSD17B10
SCHEMBL1027398 0.73 CNR2 (0.54) ALDH1A1
SCHEMBL1032165 0.73 TSHR (0.49) ALDH1A1
SCHEMBL1030344 0.73 SMN1; SMN2 (0.49) ALDH1A1MEN1KMT2AHSD17B10SMN1; SMN2
SCHEMBL1031680 0.70 HPGDS (0.48) ALDH1A1MEN1KMT2ADHODHTAS1R3
SCHEMBL4100978 0.69 ALDH1A1 (0.43) ALDH1A1MEN1KMT2AHSD17B10SMN1; SMN2
SCHEMBL1028261 0.68 TAS1R3 (0.45) ALDH1A1MEN1KMT2AHTTHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2035375-B1 1,3-DISUBSTITUTED 4-METHYL-1H-PYRROLE-2-CARBOXAMIDES AND THEIR USE FOR THE MANUFACTURE OF MEDICAMENTS GRUENENTHAL GMBH (DE) 2011-01-19 EP claimed