SCHEMBL1032473

SCHEMBL1032473

Cc1cn(Cc2ccccc2F)c(C(=O)NCCOc2ccccc2Cl)c1-c1ccc(Cl)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 7/20 0.48
NPC1 O15118 5/20 0.48
ALDH1A1 P00352 2/20 0.47
KMT2A Q03164 4/20 0.43
SMN1; SMN2 Q16637 4/20 0.43
MEN1 O00255 3/20 0.43
HPGD P15428 2/20 0.43
PKM P14618 1/20 0.43
MAPT P10636 2/20 0.40
LMNA P02545 1/20 0.40
STAT3 P40763 1/20 0.40
KLKB1 P03952 1/20 0.39
TSHR P16473 1/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
P2RX7 Q99572 1/20 0.39
HIF1A Q16665 1/20 0.38
PPARD Q03181 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1031848 0.85 RAB9A (0.53) RAB9ANPC1ALDH1A1KMT2ASMN1; SMN2
SCHEMBL1027589 0.79 MAPT (0.41) ALDH1A1KMT2ASMN1; SMN2MEN1HPGD
SCHEMBL2637921 0.78 MAPT (0.48) RAB9ANPC1ALDH1A1KMT2AMEN1
SCHEMBL1031786 0.77 PPARG (0.47) RAB9AALDH1A1HPGDPKMMAPT
SCHEMBL1029107 0.77 KDM4E (0.49) ALDH1A1KMT2ASMN1; SMN2MEN1LMNA
SCHEMBL1028192 0.73 HIF1A (0.47) RAB9ANPC1ALDH1A1KMT2AMEN1
SCHEMBL1028662 0.73 LMNA (0.48) RAB9ANPC1ALDH1A1KMT2AMEN1
SCHEMBL4103785 0.72 MAPT (0.45) RAB9ANPC1ALDH1A1KMT2ASMN1; SMN2
SCHEMBL1033737 0.71 NPC1 (0.49) RAB9ANPC1ALDH1A1KMT2ASMN1; SMN2
SCHEMBL1031268 0.69 ALDH1A1 (0.39) NPC1ALDH1A1KMT2ASMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2035375-B1 1,3-DISUBSTITUTED 4-METHYL-1H-PYRROLE-2-CARBOXAMIDES AND THEIR USE FOR THE MANUFACTURE OF MEDICAMENTS GRUENENTHAL GMBH (DE) 2011-01-19 EP claimed