SCHEMBL10366265

SCHEMBL10366265

CCn1ncc(NCCc2ccc(OC)cc2)c(Cl)c1=O

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.52
BPTF Q12830 1/20 0.52
NPBWR1 P48145 7/20 0.47
GRM2 Q14416 1/20 0.46
PDE1A P54750 1/20 0.46
PDE1B Q01064 1/20 0.46
PDE1C Q14123 1/20 0.46
CYP3A4 P08684 4/20 0.45
MCHR1 Q99705 1/20 0.44
POLB P06746 1/20 0.43
KMT2A Q03164 1/20 0.43
KDM4E B2RXH2 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MAPT P10636 2/20 0.41
BRD9 Q9H8M2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10677550 0.78 KDM4E (0.41) BRD4BPTFNPBWR1PDE1APDE1B
SCHEMBL10367314 0.78 MTNR1A (0.45) BRD4BPTFKDM4ERAB9ASMN1; SMN2
SCHEMBL9726824 0.76 PDE9A (0.49) BRD4BPTFNPBWR1CYP3A4KMT2A
SCHEMBL9726619 0.74 BRD4 (0.49) BRD4BPTFPOLBKMT2AKDM4E
SCHEMBL9726895 0.74 PDE9A (0.45) BRD4BPTFNPBWR1GRM2PDE1A
SCHEMBL10366891 0.74 SMN1; SMN2 (0.51) BRD4BPTFKMT2AKDM4ERAB9A
SCHEMBL9726665 0.73 BRD4 (0.48) BRD4BPTFCYP3A4POLBKMT2A
SCHEMBL9726673 0.71 BRD4 (0.46) BRD4BPTFPOLBKMT2AKDM4E
SCHEMBL2551062 0.71 NPBWR1 (0.77) NPBWR1CYP3A4MCHR1KMT2ARAB9A
SCHEMBL24640895 0.70 NPBWR1 (0.54) BRD4BPTFNPBWR1MCHR1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0193853-B1 3(2H)PYRIDAZINONE, PROCESS FOR ITS PREPARATION AND ANTI-ALLERGIC AGENT CONTAINING IT NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1990-09-12 EP disclosed
US-4783462-A 3(2H)pyridazinone, and anti-allergic agent containing it NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1988-11-08 US disclosed
EP-0193853-A2 3(2H)pyridazinone, process for its preparation and anti-allergic agent containing it NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1986-09-10 EP disclosed