SCHEMBL10367403

SCHEMBL10367403

OCCN1CCN(c2cc(Cl)ccc2Cl)CC1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1B P35368 11/20 0.63
HTR1A P08908 9/20 0.60
DRD2 P14416 2/20 0.59
DRD3 P35462 2/20 0.59
ADRA1A P35348 5/20 0.54
ADRA1D P25100 1/20 0.54
ALDH1A1 P00352 5/20 0.52
MAPK1 P28482 3/20 0.49
MEN1 O00255 2/20 0.49
MAPT P10636 2/20 0.49
TSHR P16473 2/20 0.49
KMT2A Q03164 2/20 0.49
NPSR1 Q6W5P4 2/20 0.49
NPC1 O15118 1/20 0.49
GMNN O75496 1/20 0.49
USP2 O75604 1/20 0.49
ABCB11 O95342 1/20 0.49
LMNA P02545 1/20 0.49
TP53 P04637 1/20 0.49
CYP1A2 P05177 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6582011 0.84 ALDH1A1 (0.73) ADRA1BHTR1ADRD3ADRA1AADRA1D
SCHEMBL11214631 0.82 ADRA1B (0.61) ADRA1BHTR1AADRA1AADRA1DUSP2
SCHEMBL9565812 0.81 DRD2 (0.79) ADRA1BHTR1ADRD2DRD3ADRA1A
SCHEMBL6580326 0.78 ADRA1B (0.72) ADRA1BHTR1AADRA1AADRA1D
SCHEMBL6577748 0.78 ADRA1B (1.00) ADRA1BHTR1AADRA1AADRA1D
SCHEMBL28513930 0.78 DRD2 (0.60) HTR1ADRD2DRD3ALDH1A1MAPT
SCHEMBL6497356 0.77 DRD2 (0.55) ADRA1BDRD2DRD3ALDH1A1MAPK1
SCHEMBL16129032 0.76 MAPT (0.62) DRD2DRD3ALDH1A1MAPK1MEN1
SCHEMBL22546968 0.76 DRD2 (0.57) ADRA1BHTR1ADRD2DRD3ADRA1A
SCHEMBL6577505 0.76 ADRA1B (0.55) ADRA1BHTR1ADRD3ADRA1AADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0094159-B1 DIHYDROPYRIDINE DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1990-03-14 EP disclosed
US-4892875-A HYPOTENSIVE, RENAL VASODILATION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1990-01-09 US disclosed
EP-0094159-A1 Dihydropyridine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1983-11-16 EP disclosed