SCHEMBL10370541

SCHEMBL10370541

O=c1[nH]c2ccsc2cc1-c1nnn[nH]1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DAO P14920 2/20 0.38
PDGFRB P09619 1/20 0.33
FGFR1 P11362 1/20 0.33
KDR P35968 1/20 0.33
CSNK2A1 P68400 1/20 0.32
TSHR P16473 2/20 0.32
KDM4E B2RXH2 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
HSD17B10 Q99714 1/20 0.31
HRH4 Q9H3N8 1/20 0.31
PDPK1 O15530 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7499608 0.75 KDR (0.60) DAOPDGFRBFGFR1KDRKDM4E
SCHEMBL10691644 0.71 DAO (0.50) DAOPDGFRBFGFR1KDR
SCHEMBL7502200 0.71 KDR (0.40) DAOPDGFRBFGFR1KDRTSHR
SCHEMBL10692085 0.71 DAO (0.52) DAOPDGFRBFGFR1KDRKDM4E
SCHEMBL7084680 0.71 KDR (0.68) PDGFRBFGFR1KDRKDM4ENPC1
Water SCHEMBL10691885 0.71 KDM4E (0.42) PDGFRBFGFR1KDRTSHRKDM4E
SCHEMBL9700418 0.69 CYP2A6 (0.34) KDM4E
SCHEMBL7503986 0.69 IDH1 (0.43) PDGFRBFGFR1KDRTSHRKDM4E
SCHEMBL10686471 0.69 KDR (0.37) DAOPDGFRBFGFR1KDRTSHR
SCHEMBL10690924 0.68 NPBWR1 (0.40) PDGFRBFGFR1KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0177924-B1 (TETRAZOLYL)THIENOPYRIDINONES MERRELL DOW PHARMACEUTICALS INC. (US) 1990-02-21 EP claimed
US-4593099-A (Tetrazolyl) thienopyridinones MERRELL DOW PHARMACEUTICALS INC. (US) 1986-06-03 US claimed
EP-0177924-A1 (Tetrazolyl)Thienopyridinones MERRELL DOW PHARMACEUTICALS INC. (US) 1986-04-16 EP claimed
EP-0177924-B1 (TETRAZOLYL)THIENOPYRIDINONES MERRELL DOW PHARMACEUTICALS INC. (US) 1990-02-21 EP disclosed
US-4593099-A (Tetrazolyl) thienopyridinones MERRELL DOW PHARMACEUTICALS INC. (US) 1986-06-03 US disclosed
EP-0177924-A1 (Tetrazolyl)Thienopyridinones MERRELL DOW PHARMACEUTICALS INC. (US) 1986-04-16 EP disclosed