SCHEMBL9700418

SCHEMBL9700418

Cc1ccsc1-c1ccc(-c2nnn[nH]2)c(=O)[nH]1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 8/20 0.34
CYP3A4 P08684 3/20 0.33
CYP2C19 P33261 3/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.33
KMT2A Q03164 1/20 0.33
CYP2B6 P20813 2/20 0.32
CYP2E1 P05181 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
PGR P06401 2/20 0.32
NISCH Q9Y2I1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9700691 0.81 PTGS2 (0.35) CYP3A4CYP2C19KDM4EMEN1ALDH1A1
SCHEMBL9700783 0.80
SCHEMBL4783148 0.77 CYP2A6 (0.46) CYP2A6CYP3A4CYP2C19KDM4EMEN1
SCHEMBL9702603 0.74
SCHEMBL9754399 0.70 MAOB (0.36) ALDH1A1
SCHEMBL9700393 0.69
SCHEMBL9702588 0.69 ALPL (0.32) ALDH1A1
SCHEMBL9700635 0.69 GAA (0.39) KDM4EMEN1ALDH1A1KMT2A
SCHEMBL10370541 0.69 DAO (0.38) KDM4E
SCHEMBL4783020 0.68 PLA2G10 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992006085-A1 PHENYLPYRIDINOL DERIVATIVES AS MEDICAMENTS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1992-04-16 WO claimed
WO-1992006085-A1 PHENYLPYRIDINOL DERIVATIVES AS MEDICAMENTS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1992-04-16 WO disclosed