SCHEMBL10380302

SCHEMBL10380302

Clc1ccc2[nH]c(C3=CC=C(c4ccc(N5CCNCC5)cc4)CC3)nc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3E A5X5Y0 3/20 0.46
HTR3B O95264 3/20 0.46
HTR3A P46098 3/20 0.46
HTR3D Q70Z44 3/20 0.46
HTR3C Q8WXA8 3/20 0.46
ADRB1 P08588 2/20 0.46
SIGMAR1 Q99720 2/20 0.46
PARP1 P09874 1/20 0.42
CETP P11597 3/20 0.42
LTA4H P09960 2/20 0.40
CHEK2 O96017 1/20 0.40
BMP4 P12644 1/20 0.39
CDC7 O00311 1/20 0.39
PIM1 P11309 1/20 0.39
CDK9 P50750 1/20 0.39
TP53 P04637 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
HTR1A P08908 1/20 0.39
CYP2D6 P10635 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10325591 0.87 HTR3E (0.51) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL1687841 0.75 HTR3E (0.54) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL19137933 0.75 RHEB (0.58) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL30489012 0.74 PARP1 (0.52) PARP1CHEK2TP53CYP3A4THRB
SCHEMBL25274071 0.74 PARP1 (0.52) PARP1CHEK2TP53CYP3A4THRB
SCHEMBL12603506 0.73 HTR3A (0.63) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL10326022 0.71 CHEK2 (0.54) CHEK2DRD2DRD3
SCHEMBL532061 0.71 ACHE (0.68) HTR3APARP1CHEK2TP53DRD2
SCHEMBL9032997 0.70 ALDH1A1 (0.62) CHEK2TP53CYP3A4HTT
SCHEMBL12101327 0.70 TOP1 (0.60) PARP1CHEK2PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012096813-A1 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-07-19 WO disclosed