SCHEMBL10388923

SCHEMBL10388923

NCC(O)c1ccc(N)c(Cl)c1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 4/20 0.40
ADRA1A P35348 4/20 0.40
ADRA2B P18089 3/20 0.40
ADRA2C P18825 3/20 0.40
ADRB2 P07550 3/20 0.40
ADRA1B P35368 2/20 0.40
CYP3A4 P08684 2/20 0.38
HSD17B10 Q99714 1/20 0.38
TAAR1 Q96RJ0 3/20 0.38
TSHR P16473 2/20 0.38
HIF1A Q16665 2/20 0.38
HTR3A P46098 1/20 0.38
NFKB1 P19838 1/20 0.38
APEX1 P27695 4/20 0.37
TDP1 Q9NUW8 4/20 0.37
KDM4E B2RXH2 3/20 0.37
MAPT P10636 3/20 0.37
RECQL P46063 3/20 0.37
BLM P54132 3/20 0.37
RAD52 P43351 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7150216 0.81 ADRA2A (0.41) ADRA2AADRA1AADRA2BADRA2CADRB2
SCHEMBL2250 0.73 ADRA2A (0.61) ADRA2AADRA1AADRA2BADRA2CADRB2
SCHEMBL21852127 0.71 ALDH1A1 (0.35) ADRA1ACYP3A4TSHRHIF1ANFKB1
SCHEMBL7147316 0.71 KCNH2 (0.54) ADRB2CYP3A4TAAR1TSHRHIF1A
SCHEMBL166818 0.71 KCNH2 (0.54) ADRB2CYP3A4TAAR1TSHRHIF1A
SCHEMBL526351 0.71 ALDH1A1 (0.50) CYP3A4HSD17B10TSHRAPEX1TDP1
SCHEMBL7149381 0.69 KIF11 (0.46) ADRA2AADRA1AADRA2BADRA2CADRB2
SCHEMBL1520565 0.68 ADRA1A (0.54) ADRA2AADRA1ATSHRNFKB1MAPT
SCHEMBL7148243 0.68 CYP3A4 (0.48) ADRA2AADRA1AADRA2BADRA2CADRB2
SCHEMBL38652517 0.67 IDO1 (0.43) ADRA2AADRA1AADRA2BADRA2CADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4906781-A Method for the preparation of 4'-(substituted)-amino-2-(substituted) amino-3',5'-dichloroacetophenone and salts thereof AMERICAN CYANAMID COMPANY (US) 1990-03-06 US disclosed