SCHEMBL2250

SCHEMBL2250

NCC(O)c1ccc(O)c(O)c1Cl

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 4/20 0.61
ADRA2B P18089 4/20 0.61
ADRA2C P18825 4/20 0.61
ADRA1A P35348 4/20 0.61
ADRB2 P07550 3/20 0.61
ADRA1B P35368 2/20 0.61
APEX1 P27695 4/20 0.46
TDP1 Q9NUW8 4/20 0.46
MAPT P10636 3/20 0.46
RECQL P46063 3/20 0.46
BLM P54132 3/20 0.46
TAAR1 Q96RJ0 3/20 0.46
KDM4E B2RXH2 3/20 0.46
HPGD P15428 2/20 0.46
CYP3A4 P08684 2/20 0.46
MEN1 O00255 1/20 0.46
LMNA P02545 1/20 0.46
ADRB1 P08588 1/20 0.46
ADORA3 P0DMS8 1/20 0.46
ADRB3 P13945 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2760850 0.78 ADRA2A (0.66) ADRA2AADRA2BADRA2CADRA1AADRB2
SCHEMBL7149381 0.76 KIF11 (0.46) ADRA2AADRA2BADRA2CADRA1AADRB2
SCHEMBL7145434 0.76 ADRA2A (0.61) ADRA2AADRA2BADRA2CADRA1AADRB2
SCHEMBL29374680 0.76 ADRA2A (1.00) ADRA2AADRA2BADRA2CADRA1AADRB2
SCHEMBL11850533 0.75 ADRB1 (0.68) ADRA2AADRA2BADRA2CADRA1AADRB2
SCHEMBL7150216 0.75 ADRA2A (0.41) ADRA2AADRA2BADRA2CADRA1AADRB2
SCHEMBL11841871 0.74 ADRB2 (0.56) ADRA2AADRA2BADRA2CADRA1AADRB2
SCHEMBL10388923 0.73 ADRA2A (0.40) ADRA2AADRA2BADRA2CADRA1AADRB2
SCHEMBL30557720 0.73 ADRA2A (0.37) ADRA2AADRA2BADRA2CADRA1AADRB2
SCHEMBL12380944 0.72 GABRA1 (0.46) ADRA2AADRA2BADRA2CADRA1AADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997030036-A1 ARYL DERIVATIVES NOVARTIS AG (CH) 1997-08-21 WO disclosed
US-5399578-A Hypotensive; valsartan; high blood pressure and cardiac insufficiency CIBA-GEIGY CORP (US) 1995-03-21 US disclosed
US-4297096-A HYPOTENSIVE AGENTS; MUSCLE RELAXANTS; STREPTOMYCES CULTURE FUJISAWA PHARMACEUTICAL CO. LTD. (JP) 1981-10-27 US disclosed