SCHEMBL10401902

SCHEMBL10401902

COc1cc(N2CCN(C(=O)NCCN(C)C)CC2)cc(OC)c1OC

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.46
GFER P55789 1/20 0.46
TP53 P04637 1/20 0.43
LMNA P02545 1/20 0.43
POLB P06746 2/20 0.42
ACVR1 Q04771 1/20 0.41
KMT2A Q03164 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
ATM Q13315 1/20 0.40
ALK Q9UM73 1/20 0.40
SUV39H2 Q9H5I1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10401560 0.99 NPC1 (0.45) NPC1GFERTP53LMNAPOLB
SCHEMBL10401512 0.87 GFER (0.58) NPC1GFERLMNAKMT2ASMN1; SMN2
Hydrochloric Acid SCHEMBL10402024 0.86 GFER (0.57) NPC1GFERLMNAKMT2ASMN1; SMN2
SCHEMBL10401976 0.81 L3MBTL1 (0.59) NPC1GFERTP53LMNAPOLB
SCHEMBL10401429 0.80 KMT2A (0.56) GFERLMNAPOLBKMT2A
SCHEMBL10401428 0.79 NPC1 (0.62) NPC1LMNA
SCHEMBL10401826 0.77 DRD2 (0.62) TP53LMNAPOLBKMT2ASMN1; SMN2
SCHEMBL10401922 0.76 MAPT (0.51) NPC1GFERTP53LMNAPOLB
SCHEMBL10401523 0.75 ALDH1A1 (0.50) NPC1GFERTP53LMNASMN1; SMN2
SCHEMBL10401849 0.75 CHRM4 (0.54) LMNAKMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4960776-A ANTIALLERGENS A. H. ROBINS COMPANY, INC. (US) 1990-10-02 US claimed
EP-0277725-A2 4-Aryl-N-[2-(dialkylamino and heterocyclicamino) alkyl]-1-piperazinecarboxamides and their use as anti allergy agents A.H. ROBINS COMPANY, INCORPORATED (US) 1988-08-10 EP claimed