SCHEMBL10401428

SCHEMBL10401428

COc1ccccc1N1CCN(C(=O)NCCN(C)C)CC1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.62
DRD2 P14416 2/20 0.60
ADRA1A P35348 1/20 0.60
DRD3 P35462 1/20 0.60
GAA P10253 2/20 0.58
L3MBTL1 Q9Y468 1/20 0.58
TSHR P16473 1/20 0.55
MAPT P10636 1/20 0.55
RAB9A P51151 1/20 0.55
LMNA P02545 1/20 0.55
HTT P42858 1/20 0.55
PKM P14618 1/20 0.54
HTR1A P08908 1/20 0.54
HTR1D P28221 1/20 0.54
HTR1B P28222 1/20 0.54
HTR2A P28223 1/20 0.54
HTR2C P28335 1/20 0.54
HTR7 P34969 1/20 0.54
HTR6 P50406 1/20 0.54
AKR1C3 P42330 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10401767 0.84 SMN1; SMN2 (0.54) NPC1DRD2DRD3GAAL3MBTL1
SCHEMBL10401740 0.83 CHRM4 (0.56) GAAL3MBTL1TSHRMAPTLMNA
Hydrochloric Acid SCHEMBL10401852 0.82 CHRM4 (0.55) GAAL3MBTL1TSHRMAPTLMNA
Hydrochloric Acid SCHEMBL10401468 0.81 CHRM4 (0.54) GAAL3MBTL1TSHRMAPTLMNA
SCHEMBL10401512 0.80 GFER (0.58) NPC1GAAL3MBTL1MAPTLMNA
SCHEMBL10401826 0.80 DRD2 (0.62) DRD2DRD3GAAMAPTLMNA
SCHEMBL5457389 0.80 DRD2 (0.73) DRD2ADRA1ADRD3DRD4
Hydrochloric Acid SCHEMBL10402024 0.79 GFER (0.57) NPC1GAAMAPTLMNAHTT
SCHEMBL10401902 0.79 NPC1 (0.46) NPC1LMNA
SCHEMBL10401976 0.78 L3MBTL1 (0.59) NPC1GAAL3MBTL1MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4960776-A ANTIALLERGENS A. H. ROBINS COMPANY, INC. (US) 1990-10-02 US claimed
EP-0277725-A2 4-Aryl-N-[2-(dialkylamino and heterocyclicamino) alkyl]-1-piperazinecarboxamides and their use as anti allergy agents A.H. ROBINS COMPANY, INCORPORATED (US) 1988-08-10 EP claimed
US-4960776-A ANTIALLERGENS A. H. ROBINS COMPANY, INC. (US) 1990-10-02 US disclosed
EP-0277725-A2 4-Aryl-N-[2-(dialkylamino and heterocyclicamino) alkyl]-1-piperazinecarboxamides and their use as anti allergy agents A.H. ROBINS COMPANY, INCORPORATED (US) 1988-08-10 EP disclosed