SCHEMBL10448709

SCHEMBL10448709

Cc1ccc(S(=O)(=O)N(C)NS(=O)(=O)c2ccccc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.56
CA9 Q16790 4/20 0.56
LMNA P02545 4/20 0.55
HTT P42858 1/20 0.55
CA2 P00918 3/20 0.53
CA1 P00915 2/20 0.53
C5AR1 P21730 1/20 0.53
ALDH1A1 P00352 6/20 0.50
GAA P10253 3/20 0.50
CYP1A2 P05177 2/20 0.50
CYP3A4 P08684 2/20 0.50
KDM4E B2RXH2 2/20 0.50
CYP2C9 P11712 2/20 0.50
CYP2C19 P33261 2/20 0.50
CYP2D6 P10635 1/20 0.50
HPGD P15428 1/20 0.50
ALOX12 P18054 1/20 0.50
GFER P55789 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
L3MBTL1 Q9Y468 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10617959 0.93 GAA (0.53) CA12CA9LMNAHTTCA2
SCHEMBL10448678 0.91 BCAT1 (0.47) CA12CA9LMNAHTTCA2
SCHEMBL10448943 0.85 ALDH1A1 (0.50) CA12CA9LMNAHTTCA2
SCHEMBL10449124 0.85 IDO1 (0.49) LMNAHTTCA2CA1ALDH1A1
SCHEMBL10449075 0.85 LMNA (0.50) CA12CA9LMNAHTTCA2
SCHEMBL10449154 0.85 EGFR (0.48) CA12CA9LMNACA2CA1
SCHEMBL10449185 0.85 LMNA (0.50) CA12CA9LMNAHTTCA2
SCHEMBL10448742 0.85 EGFR (0.48) CA12CA9LMNACA2CA1
SCHEMBL10448919 0.83 L3MBTL1 (0.59) CA12CA9LMNAHTTC5AR1
SCHEMBL10449123 0.83 ALDH1A1 (0.55) LMNACA2CA1ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4892887-A ANTITUMOR YALE UNIVERSITY (US) 1990-01-09 US disclosed
EP-0185387-B1 NOVEL, N,N'BIS(SULFONYL) HYDRAZINES HAVING ANTINEOPLASTIC ACTIVITY YALE UNIVERSITY (US) 1988-12-14 EP disclosed
US-4684747-A ANTITUMOR, ALKYLATING AGENTS YALE UNIVERSITY (US) 1987-08-04 US disclosed
EP-0185387-A1 Novel, N,N'bis(sulfonyl) hydrazines having antineoplastic activity YALE UNIVERSITY (US) 1986-06-25 EP disclosed