SCHEMBL10453021

SCHEMBL10453021

O=CCC(C(=O)O)c1ccc(CCCNS(=O)(=O)c2ccc(Cl)cc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.59
TP53 P04637 1/20 0.59
GAA P10253 1/20 0.59
TBXA2R P21731 6/20 0.53
TBXAS1 P24557 9/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
PRMT1 Q99873 2/20 0.44
AKR1C3 P42330 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10452830 0.93 TBXA2R (0.61) ALDH1A1TP53GAATBXA2RTBXAS1
SCHEMBL10453024 0.90 TBXA2R (0.58) ALDH1A1TP53GAATBXA2RTBXAS1
SCHEMBL9813854 0.84 KMT2A (0.44) ALDH1A1TP53GAATBXA2RMEN1
SCHEMBL10451941 0.83 RAB9A (0.55) ALDH1A1TBXA2RMEN1KMT2A
SCHEMBL10453042 0.83 ALDH1A1 (0.49) ALDH1A1TBXA2RTBXAS1MEN1KMT2A
SCHEMBL9813834 0.83 KMT2A (0.43) ALDH1A1TP53GAATBXA2RMEN1
SCHEMBL10452827 0.83 ALDH1A1 (0.54) ALDH1A1TBXA2RTBXAS1MEN1KMT2A
SCHEMBL10453026 0.83 TBXA2R (0.59) ALDH1A1TP53GAATBXA2RTBXAS1
SCHEMBL10452821 0.82 TAAR1 (0.57) ALDH1A1GAATBXA2RTBXAS1MEN1
SCHEMBL10451939 0.81 AKR1C3 (0.55) ALDH1A1TP53TBXA2RMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0221344-B1 SULPHONYL-PHENYL ALKYL AMINES, PROCESS FOR THEIR PREPARATION AND MEDICINES Roche Diagnostics GmbH (DE) 1990-05-23 EP disclosed