SCHEMBL10474332

SCHEMBL10474332

CSc1ccc2ccc(N)nc2n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.41
NOS2 P35228 3/20 0.35
NOS3 P29474 2/20 0.35
NOS1 P29475 1/20 0.35
BACE1 P56817 6/20 0.34
NCF1 P14598 3/20 0.34
NCK1 P16333 1/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
PLAU P00749 2/20 0.32
MCHR1 Q99705 1/20 0.32
GABRP O00591 1/20 0.31
GABRD O14764 1/20 0.31
GABRA1 P14867 1/20 0.31
GABRB1 P18505 1/20 0.31
GABRG2 P18507 1/20 0.31
GABRB3 P28472 1/20 0.31
GABRA5 P31644 1/20 0.31
GABRA3 P34903 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1765925 0.79 BACE1 (0.48) NOS2NOS3NOS1BACE1NCF1
SCHEMBL29414112 0.76 NOS2 (0.50) NOS2NOS3NOS1BACE1NCF1
SCHEMBL2901701 0.76 NOS2 (0.50) NOS2NOS3NOS1BACE1NCF1
SCHEMBL10665791 0.72 HTR7 (0.49)
SCHEMBL9376266 0.72 KDM4E (0.44) IDO1NOS2NOS3NOS1BACE1
SCHEMBL13701996 0.71
SCHEMBL6073481 0.71 HASPIN (0.41) NOS2NOS3NOS1BACE1NCF1
SCHEMBL10667360 0.70 HTR7 (0.40) NOS2NOS3NOS1KDM4EALDH1A1
SCHEMBL10754261 0.70 RAB9A (0.50) ALDH1A1LMNA
SCHEMBL6412343 0.69 PIK3CD (0.40) IDO1NOS2NOS3NOS1BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4960779-A Pyrrole derivatives, and pharmaceutical compositions which contain them and pharmacological methods of use RHONE-POULENC SANTE (FR) 1990-10-02 US disclosed
US-4642308-A ANTICONVULSANTS, ANXIOLYTIC AGENTS, ANTIEPILEPTIC AGENTS, HYPNOTICS, MUSCLE RELAXANTS RHONE-POULENC SANTE (FR) 1987-02-10 US disclosed