SCHEMBL10480368

SCHEMBL10480368

COc1c(F)cc(CNC(=S)NNC(=O)c2ccccc2)cc1F

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 6/20 0.54
CA1 P00915 1/20 0.54
CA9 Q16790 1/20 0.54
LMNA P02545 5/20 0.54
ALDH1A1 P00352 4/20 0.52
KMT2A Q03164 4/20 0.50
MEN1 O00255 3/20 0.50
ADAMTS4 O75173 1/20 0.50
ADAMTS5 Q9UNA0 1/20 0.50
ALOX12 P18054 2/20 0.49
NPC1 O15118 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
RECQL P46063 1/20 0.49
POLB P06746 1/20 0.48
MITF O75030 1/20 0.48
TDP1 Q9NUW8 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10480374 0.82 GAA (0.61) GAACA1CA9LMNAALDH1A1
SCHEMBL10480392 0.79 GAA (0.81) GAACA1CA9LMNAALDH1A1
SCHEMBL10718148 0.76 ALDH1A1 (0.39) GAAALDH1A1KMT2AMEN1
SCHEMBL31558731 0.72 KMT2A (0.72) GAACA1CA9LMNAALDH1A1
SCHEMBL6848908 0.71 SMN1; SMN2 (0.66) LMNAALDH1A1KMT2A
SCHEMBL10480438 0.71 LMNA (0.72) GAACA1CA9LMNAALDH1A1
SCHEMBL30613373 0.71 SMN1; SMN2 (0.67) LMNAALDH1A1
SCHEMBL10480431 0.71 RAB9A (0.57) GAACA1CA9LMNAALDH1A1
SCHEMBL31332476 0.70 ERCC1 (0.58) GAALMNAALDH1A1
SCHEMBL11298577 0.69 RAB9A (0.75) GAACA1CA9ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1989006125-A1 4-ARALKYL-5-SUBSTITUTED-1,2,4-TRIAZOLE-5-THIOLS SMITHKLINE BECKMAN CORPORATION (US) 1989-07-13 WO disclosed
EP-0323737-A1 4-Aralkyl-5-substituted-1,2,4-triazole-5-thiols SMITHKLINE BEECHAM CORPORATION (US) 1989-07-12 EP disclosed