SCHEMBL10480392

SCHEMBL10480392

O=C(NNC(=S)NCc1ccccc1)c1ccccc1

nearest known ligand 0.81

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GAA P10253 7/20 0.81
CA1 P00915 2/20 0.81
CA9 Q16790 2/20 0.81
ALDH1A1 P00352 3/20 0.73
MITF O75030 1/20 0.73
LMNA P02545 4/20 0.69
ADAMTS4 O75173 1/20 0.68
ADAMTS5 Q9UNA0 1/20 0.68
MEN1 O00255 1/20 0.64
KMT2A Q03164 1/20 0.64
POLB P06746 3/20 0.63
HPGD P15428 2/20 0.63
ALOX12 P18054 2/20 0.63
ALPL P05186 1/20 0.63
SMN1; SMN2 Q16637 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10480438 0.87 LMNA (0.72) GAACA1CA9ALDH1A1MITF
SCHEMBL10480374 0.85 GAA (0.61) GAACA1CA9ALDH1A1MITF
SCHEMBL14096444 0.85 ALDH1A1 (1.00) ALDH1A1MITFLMNAMEN1KMT2A
SCHEMBL9354722 0.83 TP53 (0.72) GAACA1CA9ALDH1A1MITF
SCHEMBL11374387 0.83 ALDH1A1 (0.69) GAACA1CA9ALDH1A1MITF
SCHEMBL11298577 0.82 RAB9A (0.75) GAACA1CA9ALDH1A1MEN1
SCHEMBL31558731 0.81 KMT2A (0.72) GAACA1CA9ALDH1A1LMNA
SCHEMBL457082 0.80 HDAC6 (0.79) GAAALDH1A1MITFLMNAHPGD
SCHEMBL3917581 0.79 GAA (0.68) GAACA1CA9ALDH1A1LMNA
SCHEMBL10480368 0.79 GAA (0.54) GAACA1CA9ALDH1A1MITF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1989006125-A1 4-ARALKYL-5-SUBSTITUTED-1,2,4-TRIAZOLE-5-THIOLS SMITHKLINE BECKMAN CORPORATION (US) 1989-07-13 WO disclosed
EP-0323737-A1 4-Aralkyl-5-substituted-1,2,4-triazole-5-thiols SMITHKLINE BEECHAM CORPORATION (US) 1989-07-12 EP disclosed