SCHEMBL10487828

SCHEMBL10487828

O=c1[nH]c2ccccc2c(=O)n1Cc1ccc(Cl)c(Cl)c1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 5/20 0.74
ALDH1A1 P00352 4/20 0.74
SMN1; SMN2 Q16637 3/20 0.74
KDM4E B2RXH2 2/20 0.74
TP53 P04637 2/20 0.58
MEN1 O00255 4/20 0.57
KMT2A Q03164 4/20 0.57
CYP1A2 P05177 1/20 0.55
LMNA P02545 5/20 0.55
MAPT P10636 2/20 0.55
POLB P06746 1/20 0.55
RXFP1 Q9HBX9 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
HDAC1 Q13547 1/20 0.54
TSHR P16473 1/20 0.53
MAPK10 P53779 3/20 0.52
NPSR1 Q6W5P4 2/20 0.52
HSD17B10 Q99714 2/20 0.52
USP2 O75604 1/20 0.52
HTT P42858 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10487884 0.87 ALDH1A1 (0.55) HPGDALDH1A1SMN1; SMN2KDM4ETP53
SCHEMBL6982894 0.85 HPGD (1.00) HPGDALDH1A1SMN1; SMN2KDM4ETP53
SCHEMBL30877025 0.85 HPGD (1.00) HPGDALDH1A1SMN1; SMN2KDM4ETP53
SCHEMBL10143728 0.83 LMNA (0.74) HPGDALDH1A1SMN1; SMN2KDM4ETP53
SCHEMBL17242694 0.83 KDM4E (0.50) HPGDALDH1A1SMN1; SMN2KDM4EMEN1
SCHEMBL19291210 0.82 HPGD (0.80) HPGDALDH1A1SMN1; SMN2KDM4ETP53
SCHEMBL17242542 0.80 CA12 (0.53) HPGDALDH1A1SMN1; SMN2KDM4EHDAC1
SCHEMBL7593290 0.78 MEN1 (0.77) HPGDALDH1A1SMN1; SMN2KDM4ETP53
SCHEMBL1067505 0.78 HPGD (0.78) HPGDALDH1A1SMN1; SMN2KDM4ETP53
SCHEMBL6256566 0.77 KMT2A (0.79) HPGDALDH1A1SMN1; SMN2KDM4ETP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4883800-A DIABETES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1989-11-28 US disclosed
US-4734419-A Quinazoline derivatives, compositions thereof and their use in treating diabetic complications FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1988-03-29 US disclosed
EP-0218999-A2 New quinazoline derivatives, process for their production and pharmaceutical compositions comprising them FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1987-04-22 EP disclosed