SCHEMBL10499758

SCHEMBL10499758

COc1ccc(SC(=O)c2ccc(O)cc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.50
KMT2A Q03164 3/20 0.50
ALDH1A1 P00352 3/20 0.50
ESR2 Q92731 2/20 0.50
RAB9A P51151 2/20 0.50
P4HB P07237 1/20 0.50
CALM1 P0DP23 1/20 0.50
LTA4H P09960 1/20 0.50
MEN1 O00255 1/20 0.50
F3 P13726 1/20 0.50
XDH P47989 1/20 0.50
CES2 O00748 1/20 0.50
CES1 P23141 1/20 0.50
CA1 P00915 4/20 0.48
CA2 P00918 4/20 0.48
LMNA P02545 2/20 0.48
NPC1 O15118 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
GAA P10253 1/20 0.47
PKM P14618 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL269441 0.86 ALDH1A1 (0.65) MAPTKMT2AALDH1A1RAB9ACES2
SCHEMBL1603880 0.85 MAPT (0.50) MAPTKMT2AALDH1A1ESR2RAB9A
SCHEMBL24654488 0.84 CES2 (0.59) MAPTKMT2AALDH1A1RAB9AMEN1
SCHEMBL29763732 0.84 CES2 (0.59) MAPTKMT2AALDH1A1RAB9AMEN1
SCHEMBL10499520 0.83 ELANE (0.49) MAPTKMT2AALDH1A1RAB9AMEN1
SCHEMBL10500154 0.80 LMNA (0.46) MAPTKMT2AALDH1A1CES2CES1
SCHEMBL12700321 0.77 CES2 (0.83) MAPTKMT2AALDH1A1ESR2RAB9A
SCHEMBL1817437 0.77 MAPT (0.68) MAPTKMT2AALDH1A1ESR2RAB9A
SCHEMBL19018122 0.77 MAPT (0.68) MAPTKMT2AALDH1A1ESR2RAB9A
Mequinol SCHEMBL28560858 0.77 ESR2 (0.80) KMT2AESR2RAB9ACALM1LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4849419-A 7-oxo-4-thia-azabicyclo[3,2,0]hept-2-ene derivatives HOECHST UK LIMITED (GB) 1989-07-18 US disclosed
EP-0174561-A1 7-Oxo-4-thia-1-azabicyclo[3,2,0]hept-2-ene derivatives HOECHST UK LIMITED (GB) 1986-03-19 EP disclosed
US-4131470-A THIOCARBOXYLATES VEB FILMFABRIK WOLFEN (DE) 1978-12-26 US disclosed