SCHEMBL10503271

SCHEMBL10503271

Oc1ccc(CN2CCN(CCCN3CCN(Cc4ccc(O)cc4)CC3)CC2)cc1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.56
GAA P10253 1/20 0.56
MAPT P10636 1/20 0.56
DRD4 P21917 1/20 0.54
CCR3 P51677 1/20 0.53
ESRRG P62508 2/20 0.51
MBTD1 Q05BQ5 1/20 0.50
L3MBTL3 Q96JM7 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
HRH3 Q9Y5N1 2/20 0.49
ACHE P22303 1/20 0.49
RAD52 P43351 1/20 0.49
SIGMAR1 Q99720 1/20 0.48
CACNA1G O43497 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5428090 0.89 DRD4 (0.63) ALDH1A1GAADRD4HRH3ACHE
SCHEMBL23775627 0.85 DRD4 (0.51) ALDH1A1GAAMAPTDRD4MBTD1
SCHEMBL2477654 0.84 LMNA (0.67) ALDH1A1MAPTDRD4ESRRGHRH3
SCHEMBL10502663 0.82 SIGMAR1 (0.68) ALDH1A1MAPTDRD4CCR3SIGMAR1
SCHEMBL9720752 0.82 DRD4 (0.77) GAADRD4ACHESIGMAR1
SCHEMBL9720795 0.81 CCR2 (0.54) DRD4CCR3L3MBTL1SIGMAR1
SCHEMBL322305 0.81 HRH3 (0.74) ALDH1A1DRD4MBTD1L3MBTL3L3MBTL1
SCHEMBL10502907 0.80 ALDH1A1 (0.61) ALDH1A1CCR3MBTD1L3MBTL3L3MBTL1
Hydrochloric Acid SCHEMBL10503565 0.80 SIGMAR1 (0.66) ALDH1A1MAPTDRD4CCR3SIGMAR1
SCHEMBL10686392 0.80 SIGMAR1 (0.60) MAPTCCR3SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0122488-B1 BIS-(PIPERAZINYL- OR HOMOPIPERAZINYL)-ALKANES Boehringer Ingelheim Pharmaceuticals Inc. (US) 1989-06-07 EP disclosed
US-4725597-A ANTIALLERGEN, ANTIINFLAMMATORY AGENTS BOEHRINGER INGELHEIM LTD. (US) 1988-02-16 US disclosed
EP-0122488-A1 Bis-(piperazinyl- or homopiperazinyl)-alkanes Boehringer Ingelheim Pharmaceuticals Inc. (US) 1984-10-24 EP disclosed