SCHEMBL10528043

SCHEMBL10528043

CC(=O)N(c1ccc(F)c(F)c1Cl)C1CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.43
KDM4E B2RXH2 2/20 0.37
APAF1 O14727 1/20 0.37
NPC1 O15118 1/20 0.37
TDP2 O95551 1/20 0.37
S1PR4 O95977 1/20 0.37
HSP90AA1 P07900 1/20 0.37
MAPT P10636 1/20 0.37
PKM P14618 1/20 0.37
XBP1 P17861 1/20 0.37
S1PR1 P21453 1/20 0.37
MAPK1 P28482 1/20 0.37
HTT P42858 1/20 0.37
RAB9A P51151 1/20 0.37
CACNA1B Q00975 1/20 0.37
APBA1 Q02410 1/20 0.37
PAX8 Q06710 1/20 0.37
MCL1 Q07820 1/20 0.37
HKDC1 Q2TB90 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9847870 0.73 ALDH1A1 (0.43) KDM4EAPAF1NPC1TDP2S1PR4
SCHEMBL9847843 0.71 LMNA (0.38) LMNAKDM4EAPAF1NPC1TDP2
SCHEMBL29002632 0.70 CHRM2 (0.48) LMNAKDM4EAPAF1NPC1TDP2
SCHEMBL9847891 0.70 KDM4E (0.34) KDM4ENPC1RAB9APAX8P2RX7
SCHEMBL9847871 0.70 KDM4E (0.35) LMNAKDM4EAPAF1NPC1TDP2
SCHEMBL10530512 0.69 GPR174 (0.38) LMNAKDM4EAPAF1NPC1TDP2
SCHEMBL9847821 0.68 KDM4E (0.36) LMNAKDM4EAPAF1NPC1TDP2
SCHEMBL9847872 0.67 GPR174 (0.37) LMNAKDM4ENPC1MAPTMAPK1
SCHEMBL27533046 0.66 LMNA (0.87) LMNAKDM4EAPAF1NPC1TDP2
SCHEMBL30638926 0.66 FSCN1 (0.54) NPC1MAPTRAB9AP2RX7EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1011587-B PROCESS FOR THE PREPARATION OF QUINOLONECARBOXYLIC ACID DERIVATIVES AND THEIR USE KYORIN SEIYAKU KK (JP) 1991-02-13 CN disclosed
EP-0183129-B1 QUINOLONECARBOXYLIC ACID DERIVATIVES KYORIN PHARMACEUTICAL CO., LTD. (JP) 1989-08-09 EP disclosed
CN-86102363-A The preparation method of Carbostyril carboxylic acid derivatives and application thereof 1987-01-21 CN disclosed
EP-0195841-A1 Quinolinecarboxylic acid derivatives and process for their preparation KYORIN PHARMACEUTICAL CO., LTD. (JP) 1986-10-01 EP disclosed
EP-0195316-A1 Quinolonecarboxylic acid derivatives KYORIN PHARMACEUTICAL CO., LTD. (JP) 1986-09-24 EP disclosed
CN-85109026-A The preparation method and its usage of Carbostyril carboxylic acid derivatives 1986-07-30 CN disclosed
EP-0183129-A1 Quinolonecarboxylic acid derivatives KYORIN PHARMACEUTICAL CO., LTD. (JP) 1986-06-04 EP disclosed