SCHEMBL10529751

SCHEMBL10529751

O=C(OCc1ccc([N+](=O)[O-])cc1)Oc1[c]cccc1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.53
RAB9A P51151 3/20 0.50
AKR1C3 P42330 1/20 0.46
HTT P42858 2/20 0.44
IDO1 P14902 2/20 0.43
NPC1 O15118 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10528929 0.83 ALDH1A1 (0.47) HTTTDP1L3MBTL1
SCHEMBL7867611 0.81 IDO1 (0.50) RAB9AAKR1C3IDO1NPC1
SCHEMBL6645015 0.79 RAB9A (0.61) HTR2ARAB9AAKR1C3HTTIDO1
SCHEMBL37664 0.79 HTR2A (0.62) HTR2ARAB9AAKR1C3HTTIDO1
SCHEMBL5827968 0.78 HTR2A (0.80) HTR2ARAB9AAKR1C3HTTIDO1
SCHEMBL10490876 0.77 HTR2A (0.67) HTR2ARAB9AAKR1C3HTTIDO1
SCHEMBL1714950 0.77 HTR2A (0.70) HTR2ARAB9AHTTNPC1TDP1
SCHEMBL8201751 0.77 KMT2A (0.51) TDP1
SCHEMBL10490758 0.76 HTR2A (0.58) HTR2ARAB9AAKR1C3HTTIDO1
SCHEMBL4725847 0.76 HTR2A (0.59) HTR2ARAB9AAKR1C3HTTIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0308559-A2 Cephalosporins, process for their preparation, pharmaceutical compositions containing them and intermediates BEECHAM GROUP PLC (GB) 1989-03-29 EP disclosed