SCHEMBL10568767

SCHEMBL10568767

O=C1CCc2c(OCCCN3CCN(c4ccccc4)CC3)cccc2N1CCCCc1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.58
DRD2 P14416 4/20 0.56
DRD3 P35462 4/20 0.56
DRD4 P21917 3/20 0.56
ADRB2 P07550 1/20 0.56
CHRM2 P08172 1/20 0.56
CHRM4 P08173 1/20 0.56
ADRB1 P08588 1/20 0.56
CHRM5 P08912 1/20 0.56
CHRM1 P11229 1/20 0.56
CHRM3 P20309 1/20 0.56
ADRA1D P25100 1/20 0.56
ADRA1A P35348 1/20 0.56
ADRA1B P35368 1/20 0.56
GRIN1 Q05586 1/20 0.52
GRIN2B Q13224 1/20 0.52
HTR7 P34969 3/20 0.52
HTR1A P08908 2/20 0.52
DRD5 P21918 1/20 0.52
MEN1 O00255 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10568199 0.89 SIGMAR1 (0.58) SIGMAR1DRD2DRD3DRD4ADRB2
SCHEMBL10575317 0.84 SIGMAR1 (0.54) SIGMAR1DRD2DRD3DRD4ADRB2
SCHEMBL10567416 0.84 SIGMAR1 (0.54) SIGMAR1DRD2DRD3DRD4ADRB2
SCHEMBL11065111 0.84 SIGMAR1 (0.53) SIGMAR1DRD2DRD3DRD4CHRM2
SCHEMBL10570155 0.83 HTR1A (0.57) SIGMAR1DRD2DRD3DRD4ADRB2
SCHEMBL9364940 0.82 SIGMAR1 (0.81) SIGMAR1DRD2DRD3DRD4ADRB2
SCHEMBL10569588 0.82 SIGMAR1 (0.56) SIGMAR1DRD2DRD3DRD4HTR7
Hydrochloric Acid SCHEMBL9085153 0.81 SIGMAR1 (0.80) SIGMAR1DRD2DRD3DRD4ADRB2
SCHEMBL10572966 0.79 DRD2 (0.52) SIGMAR1DRD2DRD3DRD4ADRA1D
SCHEMBL10572717 0.78 HTR1A (0.53) SIGMAR1DRD2DRD3DRD4ADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4824840-A ANTIHISTAMINES, NERVOUS SYSTEM CONTROLLERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1989-04-25 US disclosed
US-4734416-A ANTIHISTAMINES, CENTRAL NERVOUS SYSTEM CONTROLLING ACTION OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1988-03-29 US disclosed