SCHEMBL10569734

SCHEMBL10569734

N#CCc1ccccc1Cc1ccc(Br)cc1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
CSNK2A1 P68400 1/20 0.39
SLC6A2 P23975 3/20 0.38
SLC6A4 P31645 3/20 0.38
SLC6A3 Q01959 3/20 0.38
HTR2A P28223 1/20 0.36
KEAP1 Q14145 1/20 0.36
FFAR1 O14842 1/20 0.35
FFAR4 Q5NUL3 1/20 0.35
CYP1A1 P04798 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP1B1 Q16678 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MAOB P27338 2/20 0.34
TAAR1 Q96RJ0 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3636993 0.84 HTR2A (0.50) ALDH1A1HPGDSLC6A2SLC6A4SLC6A3
SCHEMBL31596156 0.84 HTR2A (0.50) ALDH1A1HPGDSLC6A2SLC6A4SLC6A3
SCHEMBL11782458 0.84 ATP4A (0.43) ALDH1A1HPGDCSNK2A1HTR2AFFAR1
SCHEMBL26988503 0.81 PYCR1 (0.42) SLC6A2SLC6A4SLC6A3HTR2AKEAP1
SCHEMBL9364439 0.81 SLC6A4 (0.41) ALDH1A1HPGDSLC6A2SLC6A4SLC6A3
SCHEMBL10566854 0.81 KEAP1 (0.58) ALDH1A1HPGDSLC6A2SLC6A4SLC6A3
SCHEMBL10564000 0.81 ALDH1A1 (0.46) ALDH1A1HPGDSLC6A2SLC6A4SLC6A3
SCHEMBL4863460 0.81 ALDH1A1 (0.41) ALDH1A1HPGDSLC6A2SLC6A4SLC6A3
SCHEMBL5703576 0.80 PYCR1 (0.45) ALDH1A1HPGDCYP1A2L3MBTL1KMT2A
SCHEMBL8763318 0.80 ALDH1A1 (0.50) ALDH1A1HPGDCSNK2A1HTR2AFFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4874763-A ANTIARRHYTHMIA AGENTS ROEHM GMBH CHEMISCHE FABRIK (DE) 1989-10-17 US disclosed
EP-0318795-A2 Pharmaceutically active pteridin derivatives Röhm GmbH (DE) 1989-06-07 EP disclosed