SCHEMBL10579477

SCHEMBL10579477

CCCCCC1C(CC(=O)O)=C(C)NC(C)=C1CC(=O)O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.39
TSHR P16473 5/20 0.39
HPGD P15428 3/20 0.39
HSD17B10 Q99714 3/20 0.39
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39
ALOX5 P09917 1/20 0.37
AKR1B1 P15121 1/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MAPT P10636 1/20 0.35
PKM P14618 1/20 0.35
FFAR3 O14843 1/20 0.34
GPR84 Q9NQS5 7/20 0.34
PPARG P37231 6/20 0.34
PPARD Q03181 6/20 0.34
PPARA Q07869 6/20 0.34
HDAC11 Q96DB2 5/20 0.34
TLR2 O60603 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2576010 0.77 LMNA (0.50) ALDH1A1TSHRHPGDHSD17B10LMNA
SCHEMBL8654462 0.76 ALDH1A1 (0.49) ALDH1A1TSHRHPGDHSD17B10LMNA
SCHEMBL8654643 0.76 ALDH1A1 (0.49) ALDH1A1TSHRHPGDHSD17B10LMNA
SCHEMBL8521929 0.74 ALDH1A1 (0.50) ALDH1A1TSHRHPGDHSD17B10LMNA
SCHEMBL8611028 0.72 ALDH1A1 (0.41) ALDH1A1TSHRHPGDHSD17B10LMNA
SCHEMBL8652188 0.72 ALDH1A1 (0.51) ALDH1A1TSHRHPGDHSD17B10LMNA
SCHEMBL7148358 0.70 ALDH1A1 (0.58) ALDH1A1TSHRHPGDHSD17B10LMNA
SCHEMBL11256668 0.69 ALDH1A1 (0.57) ALDH1A1TSHRHPGDHSD17B10LMNA
SCHEMBL2580220 0.64 ALDH1A1 (0.67) ALDH1A1HPGDLMNAMEN1KMT2A
SCHEMBL572791 0.62 ALDH1A1 (0.64) ALDH1A1HPGDLMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4868181-A CALCIUM CHANNEL BLOCKERS, ADRENERGIC BLOCKING AGENTS E. I. DU PONT DE NEMOURS AND COMPANY (US) 1989-09-19 US disclosed
EP-0255710-A2 1,4-Dihydropyridine derivatives with calcium agonist and alpha-1-antagonist activity THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1988-02-10 EP disclosed