SCHEMBL1060092

SCHEMBL1060092

CCOC(=O)CNNC(=O)OC(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
HTT P42858 1/20 0.46
CTSK P43235 2/20 0.45
GAA P10253 3/20 0.43
MGAM O43451 1/20 0.43
SI P14410 1/20 0.43
MGAM2 Q2M2H8 1/20 0.43
ALDH1A1 P00352 2/20 0.40
MEN1 O00255 1/20 0.40
TSHR P16473 1/20 0.40
KMT2A Q03164 1/20 0.40
CA12 O43570 1/20 0.39
CA2 P00918 1/20 0.39
CA14 Q9ULX7 1/20 0.39
APLNR P35414 1/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9176308 0.85 CA2 (0.43) GAAMEN1KMT2ACA12CA2
SCHEMBL7048960 0.83 CA12 (0.54) GAAMEN1TSHRKMT2ACA12
SCHEMBL1936376 0.83 ALDH1A1 (0.52) CYP1A2CYP2C9CYP2C19HTTCTSK
SCHEMBL13878757 0.83 CTSK (0.49) CYP1A2CYP2C9CYP2C19HTTCTSK
SCHEMBL7434068 0.83 GAA (0.52) CYP1A2GAAMGAMSIMGAM2
SCHEMBL402057 0.81 GAA (0.50) CYP1A2GAAMGAMSIMGAM2
SCHEMBL22660133 0.80 CTSK (0.45) CYP1A2CYP2C9CYP2C19HTTCTSK
SCHEMBL3403411 0.79 APLNR (0.49) CYP1A2CYP2C9CYP2C19HTTGAA
SCHEMBL8704463 0.78 GAA (0.44) CYP1A2CYP2C9CYP2C19HTTCTSK
SCHEMBL6355605 0.77 GAA (0.54) CYP1A2CYP2C9CYP2C19HTTCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109111371-B Preparation method of hydrazino ethyl acetate hydrochloride 江西万里药业有限公司 2021-08-06 CN claimed
WO-2011006158-A2 TARGETING NAD BIOSYNTHESIS IN BACTERIAL PATHOGENS UNIVERSITY OF MARYLAND, BALTIMORE (US) 2011-01-13 WO claimed
CN-109111371-B Preparation method of hydrazino ethyl acetate hydrochloride 江西万里药业有限公司 2021-08-06 CN disclosed
US-20190055283-A1 AZA-PEPTIDE ALDEHYDES AND KETONES OHIO STATE INNOVATION FOUNDATION 2019-02-21 US disclosed
US-8785499-B2 Targeting NAD biosynthesis in bacterial pathogens UNIVERSITY OF MARYLAND, BALTIMORE (US) 2014-07-22 US disclosed
US-8785499-B2 Targeting NAD biosynthesis in bacterial pathogens UNIVERSITY OF MARYLAND, BALTIMORE (US) 2014-07-22 US disclosed
WO-2013062881-A1 PROCESS FOR MAKING BETA 3 AGONISTS AND INTERMEDIATES MERCK SHARP & DOHME CORP. (US) 2013-05-02 WO disclosed
EP-1799653-B1 Condensed thienopyrimidine derivatives for the treatment of cancer BAYER IP GMBH (DE) 2013-03-20 EP disclosed
US-20120190708-A1 TARGETING NAD BIOSYNTHESIS IN BACTERIAL PATHOGENS UNIVERSITY OF MARYLAND, BALTIMORE (US) 2012-07-26 US disclosed
US-20120190708-A1 TARGETING NAD BIOSYNTHESIS IN BACTERIAL PATHOGENS UNIVERSITY OF MARYLAND, BALTIMORE (US) 2012-07-26 US disclosed
US-8207172-B2 Pyrimidinothienoindazoles useful for the treatment of hyperproliferative disorders BAYER INTELLECTUAL PROPERTY GMBH (DE) 2012-06-26 US disclosed
US-20110172224-A1 NOVEL HETEROCYCLES BAYER PHARMACEUTICALS CORPORATION (US) 2011-07-14 US disclosed
WO-2011006158-A2 TARGETING NAD BIOSYNTHESIS IN BACTERIAL PATHOGENS UNIVERSITY OF MARYLAND, BALTIMORE (US) 2011-01-13 WO disclosed
US-20100152098-A1 POLYBASIC BACTERIAL EFFLUX PUMP INHIBITORS AND THERAPEUTIC USES THEREOF MPEX PHARMACEUTICALS, INC. (US) 2010-06-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100152098-A1 POLYBASIC BACTERIAL EFFLUX PUMP INHIBITORS AND THERAPEUTIC USES THEREOF ABCB11, ABCB1, SLC47A1 CYP1A2 3966/4885CYP2C9 3081/4885CYP2C19 3028/4885
US-20110172224-A1 NOVEL HETEROCYCLES CCNI, PCNA, CCNA1 CYP1A2 240/4885CYP2C9 2231/4885CYP2C19 495/4885
US-20120190708-A1 TARGETING NAD BIOSYNTHESIS IN BACTERIAL PATHOGENS NAMPT, NAPRT, NADK CYP1A2 2285/4885CYP2C9 2573/4885CYP2C19 2699/4885
US-20190055283-A1 AZA-PEPTIDE ALDEHYDES AND KETONES VIP, DNPEP, PEPD CYP1A2 1714/4885CYP2C9 1546/4885CYP2C19 1112/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.