SCHEMBL10631982

SCHEMBL10631982

Fc1ccc(C(OCCN2CCN(c3c[c]ccc3)CC2)c2ccc(F)cc2)cc1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 12/20 0.73
SLC6A2 P23975 11/20 0.73
SLC6A4 P31645 11/20 0.73
SIGMAR1 Q99720 2/20 0.56
LMNA P02545 3/20 0.54
MEN1 O00255 2/20 0.54
ALDH1A1 P00352 2/20 0.54
MAPK1 P28482 2/20 0.54
KMT2A Q03164 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
TDP1 Q9NUW8 2/20 0.54
NPC1 O15118 1/20 0.54
TP53 P04637 1/20 0.54
CYP1A2 P05177 1/20 0.54
CYP3A4 P08684 1/20 0.54
CYP2D6 P10635 1/20 0.54
MAPT P10636 1/20 0.54
CYP2C9 P11712 1/20 0.54
TSHR P16473 1/20 0.54
NFKB1 P19838 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10638586 0.85 SLC6A3 (0.76) SLC6A3SLC6A2SLC6A4SIGMAR1LMNA
SCHEMBL27747290 0.83 HTR1A (0.63) SLC6A3SLC6A2SLC6A4SIGMAR1LMNA
SCHEMBL4575709 0.77 DRD2 (0.44) SLC6A3SLC6A2SLC6A4SIGMAR1MEN1
SCHEMBL597494 0.77 SLC6A3 (0.83) SLC6A3SLC6A2SLC6A4SIGMAR1LMNA
SCHEMBL8647649 0.76 LMNA (0.83) SLC6A3SLC6A2SLC6A4SIGMAR1LMNA
SCHEMBL8642037 0.76 LMNA (0.78) SLC6A3SLC6A2SLC6A4SIGMAR1LMNA
SCHEMBL8645362 0.75 LMNA (0.81) SLC6A3SLC6A2SLC6A4SIGMAR1LMNA
SCHEMBL10551886 0.75 SIGMAR1 (0.73) SLC6A3SLC6A2SLC6A4SIGMAR1LMNA
SCHEMBL9430393 0.75 SIGMAR1 (0.73) SLC6A3SLC6A2SLC6A4SIGMAR1LMNA
SCHEMBL4576039 0.75 DRD2 (0.45) SIGMAR1CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0099148-B1 PIPERAZINE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM GIST-BROCADES N.V. (NL) 1988-02-17 EP claimed
EP-0099148-B1 PIPERAZINE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM GIST-BROCADES N.V. (NL) 1988-02-17 EP disclosed